SCHEMBL9726520

SCHEMBL9726520

CCOC(=O)C(=C(c1ccc(F)cc1)c1ccc(F)cc1)c1nnn(C(C)C)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA1 P30542 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
MAPT P10636 4/20 0.38
LMNA P02545 3/20 0.38
KMT2A Q03164 3/20 0.38
NPSR1 Q6W5P4 2/20 0.38
MEN1 O00255 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
RAB9A P51151 3/20 0.37
NPC1 O15118 2/20 0.37
ELANE P08246 1/20 0.37
SLC5A1 P13866 1/20 0.37
SLC5A2 P31639 1/20 0.37
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 2/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726441 0.86 SMN1; SMN2 (0.43) SMN1; SMN2MAPTLMNAKMT2ANPSR1
SCHEMBL9726819 0.86 MAPT (0.41) ADORA2ASMN1; SMN2MAPTLMNAKMT2A
SCHEMBL9726583 0.84 SMN1; SMN2 (0.38) ADORA2AADORA3ADORA1SMN1; SMN2MAPT
SCHEMBL9726414 0.78 HMGCR (0.40) ADORA2AADORA3ADORA1SMN1; SMN2MAPT
SCHEMBL9726597 0.78 ELANE (0.39) SMN1; SMN2MAPTLMNAKMT2ANPSR1
SCHEMBL9726580 0.77 SMN1; SMN2 (0.41) SMN1; SMN2MAPTLMNAKMT2ANPSR1
SCHEMBL9726561 0.77 KDM4E (0.38) ADORA2AADORA3ADORA1SMN1; SMN2MAPT
SCHEMBL9726678 0.77 HMGCR (0.38) ADORA2AADORA3ADORA1SMN1; SMN2LMNA
SCHEMBL9726424 0.76 HMGCR (0.36) ADORA2AADORA3ADORA1SMN1; SMN2RAB9A
SCHEMBL9726560 0.74 HMGCR (0.44) ADORA2AADORA3ADORA1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
US-4897490-A DERIVATIVES OF BETA-HYDROXY,OMEGA-DIPHENYL,TETRAZOL-5-YL ALK-OMEGA-ENOIC ACID, ESTER OR LACTONE BRISTOL-MEYERS COMPANY (US) 1990-01-30 US disclosed
WO-1988006584-A1 ANTIHYPERCHOLESTEROLEMIC TETRAZOLE COMPOUNDS BRISTOL-MYERS COMPANY (US) 1988-09-07 WO disclosed