SCHEMBL9726424

SCHEMBL9726424

CC(C)n1nnc(C(C=O)=C(c2ccc(F)cc2)c2ccc(F)cc2)n1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 2/20 0.36
ATM Q13315 1/20 0.32
ADORA2A P29274 2/20 0.32
ADORA1 P30542 2/20 0.32
RAB9A P51151 3/20 0.31
NPC1 O15118 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
MGLL Q99685 1/20 0.30
ADORA3 P0DMS8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726747 0.88 HMGCR (0.36) HMGCR
SCHEMBL9726752 0.88 HMGCR (0.36) HMGCR
SCHEMBL9726434 0.83 HSD11B1 (0.37) HMGCRATMRAB9ANPC1SMN1; SMN2
SCHEMBL9726796 0.82 HMGCR (0.32) HMGCRRAB9ASMN1; SMN2
SCHEMBL9726403 0.82 TRPM8 (0.42) HMGCRRAB9ANPC1SMN1; SMN2
SCHEMBL10608830 0.76 TRPA1 (0.34)
SCHEMBL9726520 0.76 ADORA2A (0.39) ADORA2AADORA1RAB9ANPC1SMN1; SMN2
SCHEMBL10611915 0.76 HMGCR (0.57) HMGCR
SCHEMBL9726484 0.75 HMGCR (0.43) HMGCR
SCHEMBL9726567 0.74 HMGCR (0.44) HMGCRADORA2AADORA1SMN1; SMN2ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110940-A Inhibitors of 3-hydroxy-3-methylglutaryl coenzyme A reductase BRISTOL-MYERS COMPANY (US) 1992-05-05 US disclosed
US-5068346-A Anticholesterol agents BRISTOL-MYERS COMPANY (US) 1991-11-26 US disclosed
US-4897490-A DERIVATIVES OF BETA-HYDROXY,OMEGA-DIPHENYL,TETRAZOL-5-YL ALK-OMEGA-ENOIC ACID, ESTER OR LACTONE BRISTOL-MEYERS COMPANY (US) 1990-01-30 US disclosed
WO-1988006584-A1 ANTIHYPERCHOLESTEROLEMIC TETRAZOLE COMPOUNDS BRISTOL-MYERS COMPANY (US) 1988-09-07 WO disclosed