SCHEMBL9726950

SCHEMBL9726950

O=C1NCCCC12CCCN(C(c1ccccc1)c1ccccc1)C2=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 2/20 0.43
GRIN2A Q12879 2/20 0.43
USP2 O75604 6/20 0.40
CYP3A4 P08684 5/20 0.40
CYP2D6 P10635 5/20 0.40
CYP1A2 P05177 3/20 0.40
TP53 P04637 1/20 0.40
ALOX15 P16050 1/20 0.40
OPRM1 P35372 7/20 0.40
OPRD1 P41143 7/20 0.40
OPRK1 P41145 7/20 0.40
OPRL1 P41146 7/20 0.40
CYP2C9 P11712 5/20 0.39
ALDH1A1 P00352 1/20 0.39
GRIN2B Q13224 1/20 0.38
CYP2C19 P33261 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
RAB9A P51151 1/20 0.34
TSHR P16473 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727040 0.85 MEN1 (0.49) USP2CYP3A4CYP2D6CYP1A2TP53
SCHEMBL19341589 0.75 USP2 (0.51) USP2CYP3A4CYP2D6CYP1A2TP53
SCHEMBL9726828 0.73 KMT2A (0.74) GRIN1GRIN2ACYP2D6OPRM1OPRD1
SCHEMBL19341586 0.72 OPRM1 (0.53) GRIN1GRIN2AUSP2CYP3A4CYP2D6
SCHEMBL5563143 0.68 KMT2A (0.48) USP2CYP3A4CYP2D6CYP1A2OPRM1
SCHEMBL19347109 0.68 CYP3A4 (0.56) USP2CYP3A4CYP2D6CYP1A2TP53
SCHEMBL9726922 0.66 GRIN1 (0.38) GRIN1GRIN2AGRIN2B
SCHEMBL7043309 0.65 GRIN1 (0.42) GRIN1GRIN2AUSP2CYP3A4CYP2D6
SCHEMBL7043301 0.65 GRIN1 (0.41) GRIN1GRIN2AUSP2CYP3A4CYP2D6
SCHEMBL6730231 0.63 GRIN1 (0.40) GRIN1GRIN2AOPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5128466-A For monitoring lithium levels in patients receiving lithium treatment for depression THE RESEARCH FOUNDATION OF STATE UNIVERSITY OF NEW YORK (US) 1992-07-07 US disclosed