SCHEMBL9727207

SCHEMBL9727207

COc1cccc2c1CC(N1CCC1)CC2

nearest known ligand 0.92

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.55
CHRM1 P11229 2/20 0.55
CHRM3 P20309 2/20 0.55
SIGMAR1 Q99720 1/20 0.52
MTNR1A P48039 1/20 0.49
MTNR1B P49286 1/20 0.49
DRD2 P14416 2/20 0.49
DRD3 P35462 2/20 0.49
HTR2C P28335 1/20 0.48
HTR2B P41595 1/20 0.48
DRD1 P21728 1/20 0.48
DRD5 P21918 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4215401 0.97 CHRM2 (0.55) CHRM2CHRM1CHRM3SIGMAR1MTNR1A
SCHEMBL11393302 0.96 SIGMAR1 (0.54) CHRM2CHRM1CHRM3SIGMAR1MTNR1A
SCHEMBL8677765 0.96 SIGMAR1 (0.54) CHRM2CHRM1CHRM3SIGMAR1MTNR1A
Hydrochloric Acid SCHEMBL7933015 0.94 SIGMAR1 (0.53) CHRM2CHRM1CHRM3SIGMAR1MTNR1A
Hydrochloric Acid SCHEMBL7935858 0.94 SIGMAR1 (0.53) CHRM2CHRM1CHRM3SIGMAR1MTNR1A
SCHEMBL9239027 0.90 DRD2 (0.54) CHRM2CHRM1CHRM3SIGMAR1DRD2
Hydrochloric Acid SCHEMBL9243515 0.89 DRD2 (0.52) CHRM2CHRM1CHRM3SIGMAR1DRD2
Hydrochloric Acid SCHEMBL9242362 0.89 DRD2 (0.52) CHRM2CHRM1CHRM3SIGMAR1DRD2
SCHEMBL8674841 0.89 CHRM2 (0.56) CHRM2CHRM1CHRM3SIGMAR1MTNR1A
Hydrochloric Acid SCHEMBL7932854 0.87 CHRM2 (0.55) CHRM2CHRM1CHRM3SIGMAR1MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164385-A AZETIDINE DERIVATIVES AND HYPOTENSIVE COMPOSITIONS THEREOF JOHN WYETH & BROTHER, LTD. (GB) 1992-11-17 US claimed
US-5164385-A AZETIDINE DERIVATIVES AND HYPOTENSIVE COMPOSITIONS THEREOF JOHN WYETH & BROTHER, LTD. (GB) 1992-11-17 US disclosed