SCHEMBL9727328

SCHEMBL9727328

O=S(=O)(Cl)c1ccc(C2CCCCCN2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C19 P33261 2/20 0.47
CHRNB2 P17787 2/20 0.47
CHRNA7 P36544 2/20 0.47
CHRNA4 P43681 2/20 0.47
POLB P06746 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2A6 P11509 1/20 0.47
CYP2C9 P11712 1/20 0.47
AURKA O14965 1/20 0.41
MKNK1 Q9BUB5 1/20 0.40
PARP1 P09874 4/20 0.39
PARP2 Q9UGN5 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
MAPKAPK2 P49137 1/20 0.37
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16401187 0.82 KMT2A (0.45) KMT2AMEN1CYP2D6CYP2C19CHRNB2
SCHEMBL16400474 0.82 CA2 (0.45) KMT2AMEN1CYP2D6CYP2C19CHRNB2
SCHEMBL16409298 0.78 SMN1; SMN2 (0.43) KMT2AMEN1CYP2D6CYP2C19CHRNB2
SCHEMBL24313467 0.78 MEN1 (0.50) KMT2AMEN1CYP2D6CYP2C19CHRNB2
SCHEMBL21962249 0.77 CHRNA7 (0.44) KMT2AMEN1CYP2D6CYP2C19CHRNB2
SCHEMBL28307604 0.77 MKNK1 (0.49) KMT2AMEN1CYP2D6CYP2C19CHRNB2
Acetic Acid SCHEMBL27869895 0.76 KMT2A (0.43) KMT2AMEN1CYP2D6CYP2C19CHRNB2
SCHEMBL11677845 0.75 LMNA (0.59) KMT2AMEN1CHRNA7POLBSMN1; SMN2
SCHEMBL29347914 0.75 MEN1 (0.51) KMT2AMEN1CYP2D6CYP2C19CHRNB2
SCHEMBL1931626 0.75 LMNA (0.59) KMT2AMEN1CHRNA7POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164514-A Antispasmodics ROUSSEL UCLAF (FR) 1992-11-17 US disclosed
US-5081130-A Antispasmodic agents ROUSSEL UCLAF (FR) 1992-01-14 US disclosed
US-5041436-A 1-arylsulphonyl-2-piperidinone derivatives, process and intermediates for the preparation thereof, their application as antispasmodics and compositions containing them ROUSSEL UCLAF (FR) 1991-08-20 US disclosed
US-5037822-A Antispasmodic agent ROUSSEL-UCLAF (FR) 1991-08-06 US disclosed
US-4990531-A Antispasmodic agents ROUSSEL UCLAF (FR) 1991-02-05 US disclosed