SCHEMBL9727330

SCHEMBL9727330

O=S(=O)(Cl)c1ccccc1C1CCCNCC1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 9/20 0.46
HTR2C P28335 8/20 0.46
HTR1A P08908 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
SLC18A3 Q16572 1/20 0.40
SIGMAR1 Q99720 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9865925 0.95 HTR6 (0.45) HTR6HTR2CHTR1ASLC6A2SLC6A4
SCHEMBL9727510 0.94 HTR2C (0.51) HTR6HTR2CHTR1ASLC6A2SLC6A4
SCHEMBL9732296 0.84 HTR6 (0.42) HTR6HTR2C
SCHEMBL9727253 0.84 PTGS2 (0.46)
SCHEMBL23045663 0.82 HSD11B1 (0.44) HTR6HTR2C
SCHEMBL6606000 0.78 HTR2C (0.56) HTR6HTR2CHTR1ASLC6A2SLC6A4
SCHEMBL4623351 0.78 HTR2C (0.51) HTR6HTR2CHTR1ASLC6A2SLC6A4
SCHEMBL29764435 0.78 HTR2C (0.51) HTR6HTR2CHTR1ASLC6A2SLC6A4
Hydrochloric Acid SCHEMBL4891683 0.76 HTR2C (0.57) HTR6HTR2CHTR1ASLC6A2SLC6A4
SCHEMBL7819186 0.74 HTR2C (0.51) HTR6HTR2CHTR1ASLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164514-A Antispasmodics ROUSSEL UCLAF (FR) 1992-11-17 US disclosed
US-5081130-A Antispasmodic agents ROUSSEL UCLAF (FR) 1992-01-14 US disclosed
US-5041436-A 1-arylsulphonyl-2-piperidinone derivatives, process and intermediates for the preparation thereof, their application as antispasmodics and compositions containing them ROUSSEL UCLAF (FR) 1991-08-20 US disclosed
US-5037822-A Antispasmodic agent ROUSSEL-UCLAF (FR) 1991-08-06 US disclosed
US-4990531-A Antispasmodic agents ROUSSEL UCLAF (FR) 1991-02-05 US disclosed