SCHEMBL9727341

SCHEMBL9727341

CCCN(CCC)c1ccc(S(=O)(=O)Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.42
ERBB2 P04626 2/20 0.42
RORC P51449 3/20 0.40
ALDH1A1 P00352 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
HSD17B10 Q99714 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40
CNR2 P34972 6/20 0.39
CNR1 P21554 2/20 0.39
ESR1 P03372 1/20 0.38
CA12 O43570 1/20 0.38
CA2 P00918 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CA9 Q16790 1/20 0.38
SLC22A6 Q4U2R8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11769284 0.93 ALDH1A1 (0.45) ALDH1A1L3MBTL1MEN1MAPTHPGD
SCHEMBL9727371 0.89 EGFR (0.45) EGFRERBB2ALDH1A1TDP1HSD17B10
SCHEMBL3223255 0.84 ALDH1A1 (0.55) ALDH1A1TDP1L3MBTL1MEN1MAPT
SCHEMBL3225090 0.82 CNR2 (0.48) EGFRERBB2ALDH1A1TDP1HSD17B10
SCHEMBL414561 0.81 CA2 (0.56) ALDH1A1TDP1MEN1KMT2ACA12
SCHEMBL4224314 0.79 EGFR (0.44) EGFRERBB2ALDH1A1TDP1L3MBTL1
SCHEMBL23363660 0.78 ALDH1A1 (0.41) ALDH1A1TDP1HSD17B10L3MBTL1MEN1
SCHEMBL7150414 0.78 EGFR (0.47) EGFRERBB2ALDH1A1TDP1L3MBTL1
SCHEMBL24763419 0.76 ESR1 (0.42) ALDH1A1HSD17B10MAPTKMT2ACNR2
SCHEMBL28264310 0.75 ENPP2 (0.41) EGFRERBB2RORCALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164514-A Antispasmodics ROUSSEL UCLAF (FR) 1992-11-17 US disclosed
US-5081130-A Antispasmodic agents ROUSSEL UCLAF (FR) 1992-01-14 US disclosed
US-5041436-A 1-arylsulphonyl-2-piperidinone derivatives, process and intermediates for the preparation thereof, their application as antispasmodics and compositions containing them ROUSSEL UCLAF (FR) 1991-08-20 US disclosed
US-4990531-A Antispasmodic agents ROUSSEL UCLAF (FR) 1991-02-05 US disclosed