SCHEMBL9727746

SCHEMBL9727746

C=CCc1cc2c(cc1O)C(C)(C)C(OC)O2

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.36
GABRB2 P47870 1/20 0.36
PTPN1 P18031 5/20 0.34
SRD5A1 P18405 1/20 0.34
CYP3A4 P08684 2/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B1 P14061 1/20 0.32
POLB P06746 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ALOX5 P09917 1/20 0.32
AR P10275 1/20 0.32
PTGS1 P23219 1/20 0.32
TRPM8 Q7Z2W7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9727666 0.82 GABRA1 (0.38) GABRA1GABRB2PTPN1SRD5A1HSD17B1
SCHEMBL9727754 0.78 GABRA1 (0.35) GABRA1GABRB2PTPN1SRD5A1HSD17B1
SCHEMBL9727707 0.74 PTPN1 (0.37) PTPN1SRD5A1
SCHEMBL9727784 0.71 SRD5A1 (0.35) GABRA1GABRB2SRD5A1CYP3A4ALDH1A1
SCHEMBL1420694 0.65 GABRA1 (0.64) GABRA1GABRB2PTPN1SRD5A1CYP3A4
SCHEMBL1276635 0.65 CYP3A4 (0.55) GABRA1GABRB2PTPN1SRD5A1CYP3A4
SCHEMBL13387030 0.64 HMGCR (0.56) GABRA1GABRB2PTPN1CYP3A4ALOX15
SCHEMBL6309438 0.63 GABRA1 (0.61) GABRA1GABRB2PTPN1SRD5A1CYP3A4
SCHEMBL15269320 0.62 CYP3A4 (0.57) GABRA1GABRB2PTPN1CYP3A4ALOX15
SCHEMBL9727708 0.62 ALDH1A1 (0.42) GABRA1GABRB2PTPN1CYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5091533-A Treating allergies, cardiovascular disorders, inflammation MERCK FROSST CANADA, INC. (CA) 1992-02-25 US disclosed
EP-0447189-A1 5-Hydroxy-2,3-dihydrobenzofuran analogs as leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1991-09-18 EP disclosed