SCHEMBL9729303

SCHEMBL9729303

c1c[nH]c2cc3cncc3cc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.40
PIK3CB P42338 1/20 0.40
PIK3CG P48736 1/20 0.40
FYN P06241 1/20 0.38
GPR84 Q9NQS5 1/20 0.38
NPC1 O15118 1/20 0.37
TRPA1 O75762 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
ITGB2 P05107 1/20 0.37
ICAM1 P05362 1/20 0.37
ITGAL P20701 1/20 0.37
CA4 P22748 1/20 0.37
CA6 P23280 1/20 0.37
AHR P35869 1/20 0.37
ADK P55263 1/20 0.37
CYP19A1 P11511 1/20 0.36
HASPIN Q8TF76 4/20 0.36
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11172742 0.98 PIK3CD (0.39) PIK3CDPIK3CBPIK3CGFYNGPR84
Maleic Acid SCHEMBL11162454 0.85 CCNC (0.44) HASPINCCNT1CDK9
SCHEMBL2806310 0.82 GPR84 (0.43) GPR84NPC1TRPA1CA1CA2
SCHEMBL16241832 0.76 HASPIN (0.51) PIK3CDPIK3CBPIK3CGGPR84HASPIN
SCHEMBL7493615 0.76 HASPIN (0.51) PIK3CDPIK3CBPIK3CGGPR84HASPIN
Hydrochloric Acid SCHEMBL8560372 0.75 HASPIN (0.50) PIK3CDPIK3CBPIK3CGGPR84HASPIN
SCHEMBL30071614 0.73 AHR (0.61) GPR84NPC1TRPA1CA1CA2
SCHEMBL1440181 0.73 AHR (0.61) GPR84NPC1TRPA1CA1CA2
SCHEMBL6151694 0.72 ALDH1A1 (0.50) FYNGPR84NPC1TRPA1CA1
Hydrochloric Acid SCHEMBL7763064 0.71 AHR (0.58) GPR84NPC1TRPA1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0250179-A2 BCD tricyclic ergoline part-structure analogues ELI LILLY AND COMPANY (US) 1987-12-23 EP claimed
EP-0013788-B1 OCTAHYDRO-2H-PYRROLO(3,4-G)QUINOLINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ELI LILLY AND COMPANY (US) 1983-04-27 EP claimed
US-5134143-A Dopamine Agonists ELI LILLY AND COMPANY (US) 1992-07-28 US disclosed
US-5134143-A Dopamine Agonists ELI LILLY AND COMPANY (US) 1992-07-28 US disclosed
CN-1016872-B BCD TRICYCLIC ERGOLINE PART-STRUCTURE ANALOGUSE LILLY CO ELI (US) 1992-06-03 CN disclosed
US-4977160-A DOPAMINE AGONISTS; PARKINSON*S DISEASE ELI LILLY AND COMPANY (US) 1990-12-11 US disclosed
US-4977160-A DOPAMINE AGONISTS; PARKINSON*S DISEASE ELI LILLY AND COMPANY (US) 1990-12-11 US disclosed
US-4826986-A DOPAMINE AGONISTS ELI LILLY AND COMPANY (US) 1989-05-02 US disclosed
US-4826986-A DOPAMINE AGONISTS ELI LILLY AND COMPANY (US) 1989-05-02 US disclosed
EP-0250179-A2 BCD tricyclic ergoline part-structure analogues ELI LILLY AND COMPANY (US) 1987-12-23 EP disclosed
EP-0250179-A2 BCD tricyclic ergoline part-structure analogues ELI LILLY AND COMPANY (US) 1987-12-23 EP disclosed
EP-0142920-A2 6-Oxodecahydroquinolines and process for their preparation ELI LILLY AND COMPANY (US) 1985-05-29 EP disclosed
EP-0013788-B1 OCTAHYDRO-2H-PYRROLO(3,4-G)QUINOLINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ELI LILLY AND COMPANY (US) 1983-04-27 EP disclosed
US-4311844-A Octahydro-2H-pyrrolo[3,4,-g]quinolines ELI LILLY AND COMPANY (US) 1982-01-19 US disclosed
US-4282362-A TREATING PARKINSON'S DISEASE, INHIBITORS OF PRE ACTIN SECRETION, DOPAMINE ANTAGONISTS ELI LILLY AND COMPANY (US) 1981-08-04 US disclosed
US-4235909-A DOPAMINE ANTAGONISTS, IN THE TREATMENT OF PARKINSON'S DISEASE ELI LILLY AND COMPANY (US) 1980-11-25 US disclosed
EP-0013788-A1 Octahydro-2H-pyrrolo(3,4-g)quinolines, process for their preparation and pharmaceutical compositions containing them ELI LILLY AND COMPANY (US) 1980-08-06 EP disclosed