SCHEMBL9729305

SCHEMBL9729305

CC(C)c1cccc(C(C)C)c1-n1nnn(CC(C)(C)C)c1=S

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.37
ALDH1A1 P00352 1/20 0.37
ALOX15 P16050 1/20 0.37
DPP4 P27487 3/20 0.36
ANPEP P15144 2/20 0.36
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
GABRA1 P14867 2/20 0.31
GABRG2 P18507 2/20 0.31
GABRB3 P28472 2/20 0.31
FAAH O00519 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
LMNA P02545 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
HPGD P15428 1/20 0.30
GABRB1 P18505 1/20 0.30
PTGS1 P23219 1/20 0.30
SLC6A2 P23975 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9728711 0.93 TSHR (0.46) TSHRALDH1A1ALOX15DPP4ANPEP
SCHEMBL9728430 0.90 DPP4 (0.33) TSHRALDH1A1ALOX15DPP4ANPEP
SCHEMBL9728613 0.77 GABRA1 (0.37) TSHRALDH1A1GABRA1CA2CYP3A4
SCHEMBL9728180 0.74 DPP4 (0.42) TSHRALDH1A1ALOX15DPP4ANPEP
SCHEMBL9728307 0.70 TSHR (0.50) TSHRALDH1A1ALOX15DPP4ANPEP
SCHEMBL9728387 0.69 DPP4 (0.36) TSHRALDH1A1ALOX15DPP4ANPEP
SCHEMBL9728918 0.69 ALDH1A1 (0.46) TSHRALDH1A1ALOX15DPP4ANPEP
SCHEMBL9728241 0.68 DPP4 (0.37) TSHRALDH1A1ALOX15DPP4ANPEP
SCHEMBL9728643 0.67 DPP4 (0.39) TSHRALDH1A1ALOX15DPP4ANPEP
SCHEMBL9728513 0.66 TSHR (0.36) TSHRALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0406163-A1 Thioxotetrazolines CIBA-GEIGY AG (CH) 1991-01-02 EP claimed
US-5138068-A Pesticide CIBA-GEIGY CORPORATION (US) 1992-08-11 US disclosed
US-5066667-A Controlling insects and arachnids CIBA-GEIGY CORPORATION (US) 1991-11-19 US disclosed
EP-0406163-A1 Thioxotetrazolines CIBA-GEIGY AG (CH) 1991-01-02 EP disclosed