SCHEMBL9731103

SCHEMBL9731103

NC(=O)NC(=O)c1ccc2ccccc2c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 4/20 0.58
DEGS1 O15121 1/20 0.58
NPC1 O15118 6/20 0.57
RAB9A P51151 6/20 0.57
KDM4E B2RXH2 2/20 0.57
CES2 O00748 1/20 0.57
CES1 P23141 1/20 0.57
F2 P00734 2/20 0.55
PLG P00747 2/20 0.55
KLKB1 P03952 2/20 0.55
KLK1 P06870 2/20 0.55
PRSS1 P07477 2/20 0.55
PLAT P00750 1/20 0.55
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
CASP3 P42574 1/20 0.54
SENP7 Q9BQF6 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
HDAC3 O15379 1/20 0.51
HDAC1 Q13547 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8161115 0.89 NPC1 (0.62) PLAUDEGS1NPC1RAB9AKDM4E
SCHEMBL5430957 0.86 PLAU (0.59) PLAUDEGS1NPC1RAB9AKDM4E
Hydrochloric Acid SCHEMBL8700251 0.84 PLAU (0.58) PLAUDEGS1NPC1RAB9AKDM4E
Guanidine SCHEMBL27709689 0.84 PLAU (0.58) PLAUDEGS1NPC1RAB9AKDM4E
SCHEMBL6010047 0.84 F12 (0.55) PLAUDEGS1NPC1RAB9AF2
SCHEMBL8009175 0.83 NPC1 (0.59) PLAUDEGS1NPC1RAB9AKDM4E
SCHEMBL5432538 0.81 CES2 (0.57) PLAUDEGS1NPC1RAB9AKDM4E
SCHEMBL27373888 0.81 NPC1 (0.58) DEGS1NPC1RAB9AKDM4ECES2
SCHEMBL1149678 0.81 NPC1 (0.62) DEGS1NPC1RAB9AKDM4ECES2
Naphthalene SCHEMBL27966015 0.81 ALDH1A1 (0.60) NPC1RAB9AMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5106843-A Treatment of migraine, emesis, anxiety, gastrointestinal disorders, psychological disorders AMERICAN HOME PRODUCTS CORPORATION (US) 1992-04-21 US disclosed
EP-0323077-B1 HETEROCYCLIC COMPOUNDS JOHN WYETH & BROTHER LIMITED (GB) 1991-09-11 EP disclosed
US-4983600-A Antiemetics, antianxiety agents, gastrointestinal disorders JOHN WYETH & BROTHER LIMITED (GB) 1991-01-08 US disclosed
EP-0323077-A1 Heterocyclic compounds JOHN WYETH & BROTHER LIMITED (GB) 1989-07-05 EP disclosed