SCHEMBL9733201

SCHEMBL9733201

C#CCC(CCCC#N)CCC(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.40
CYP2D6 P10635 2/20 0.40
MAPT P10636 2/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HSD17B10 Q99714 1/20 0.40
NFKB1 P19838 1/20 0.39
LMNA P02545 1/20 0.39
GSTK1 Q9Y2Q3 2/20 0.34
TSHR P16473 1/20 0.33
SLC1A2 P43004 2/20 0.32
TET2 Q6N021 3/20 0.31
KDM4A O75164 2/20 0.31
KDM4C Q9H3R0 2/20 0.31
KDM2A Q9Y2K7 2/20 0.31
TET3 O43151 1/20 0.31
GABRP O00591 2/20 0.31
GABRD O14764 2/20 0.31
GABRA1 P14867 2/20 0.31
GABRB1 P18505 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16085876 0.76 CYP2D6 (0.45) CYP1A2CYP2D6MAPTCYP2C9CYP2C19
SCHEMBL9732893 0.75 MAPT (0.39) CYP1A2CYP2D6MAPTCYP2C9CYP2C19
SCHEMBL23848 0.70
SCHEMBL454017 0.68
Adipic Acid SCHEMBL28268122 0.68 LMNA (0.58) CYP1A2CYP2D6MAPTCYP2C9CYP2C19
Adipic Acid SCHEMBL9504707 0.68 LMNA (0.58) CYP1A2CYP2D6MAPTCYP2C9CYP2C19
Ammonia Solution, Strong SCHEMBL5709311 0.68
SCHEMBL17935639 0.68 TSHR (0.42) MAPTTSHR
SCHEMBL3761638 0.66 TSHR (0.60) CYP1A2CYP2D6MAPTCYP2C9CYP2C19
SCHEMBL609292 0.66 TSHR (0.60) CYP1A2CYP2D6MAPTCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5153214-A Treating cardiovascular disorders CIBA-GEIGY CORPORATION (US) 1992-10-06 US disclosed
US-5025025-A Cardiovascular disorders CIBA-GEIGY CORPORATION (US) 1991-06-18 US disclosed
EP-0405391-A1 Certain (arylsulfonamido- and pyridyl- or imidazolyl-)-substituted carboxylic acids and derivatives thereof CIBA-GEIGY AG (CH) 1991-01-02 EP disclosed