SCHEMBL9733229

SCHEMBL9733229

CC1(C)C=C(n2cc([N+](=O)[O-])cc([N+](=O)[O-])c2=O)c2cc(C#N)ccc2C1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 2/20 0.35
ALK Q9UM73 1/20 0.34
ABCC9 O60706 1/20 0.34
MAPT P10636 3/20 0.34
MAPK1 P28482 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
KCNJ1 P48048 2/20 0.33
KCNH2 Q12809 2/20 0.33
AR P10275 1/20 0.31
KMT2A Q03164 2/20 0.31
DGKI O75912 1/20 0.31
DGKA P23743 1/20 0.31
DGKZ Q13574 1/20 0.31
MEN1 O00255 1/20 0.30
ESRRA P11474 1/20 0.30
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733247 0.90 VCAM1 (0.39) VCAM1ALKABCC9MAPTMAPK1
SCHEMBL9733596 0.90 VCAM1 (0.34) VCAM1ALKABCC9MAPTMAPK1
SCHEMBL9733168 0.89 ABCC9 (0.34) VCAM1ALKABCC9KCNJ1KCNH2
SCHEMBL9733591 0.89 VCAM1 (0.37) VCAM1ALKABCC9KCNJ1KCNH2
SCHEMBL9733088 0.86 MAPT (0.36) VCAM1ALKABCC9MAPTMAPK1
SCHEMBL9733322 0.86 KCNJ1 (0.36) VCAM1ALKABCC9MAPTMAPK1
SCHEMBL8088704 0.80 ABCC9 (0.40) VCAM1ABCC9MAPTMAPK1TDP1
SCHEMBL9734810 0.77 ABCC9 (0.32) ABCC9
SCHEMBL9733508 0.77 PGR (0.32) ALK
SCHEMBL9734137 0.76 BACE1 (0.35) ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP disclosed