SCHEMBL9733979

SCHEMBL9733979

CC(C)c1cc(CN2CCCN(Cc3cc(C(C)C)cc(C(C)C)c3O)C2)c(O)c(C(C)C)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
GABRA1 P14867 1/20 0.45
GABRB2 P47870 1/20 0.45
KDM4E B2RXH2 2/20 0.43
MPO P05164 1/20 0.43
MAPT P10636 2/20 0.41
TSHR P16473 3/20 0.39
ALDH1A1 P00352 3/20 0.39
LMNA P02545 2/20 0.39
FABP3 P05413 2/20 0.36
FABP4 P15090 2/20 0.36
FABP5 Q01469 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
ALOX15 P16050 1/20 0.35
HIF1A Q16665 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MEN1 O00255 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733841 0.93 MAPT (0.52) MAPK1CYP1A2CYP2D6GABRA1GABRB2
SCHEMBL9736352 0.90 MAPK1 (0.44) MAPK1CYP1A2CYP2D6GABRA1GABRB2
SCHEMBL9734778 0.85 MAPK1 (0.49) MAPK1CYP1A2CYP2D6KDM4EMPO
SCHEMBL9733983 0.78 MAPT (0.65) MAPK1CYP1A2CYP2D6GABRA1GABRB2
SCHEMBL8897499 0.77 GABRA1 (0.61) CYP1A2CYP2D6GABRA1GABRB2TSHR
SCHEMBL9734442 0.73 MAPT (0.55) MAPK1CYP1A2CYP2D6GABRA1GABRB2
SCHEMBL14682849 0.72 GABRA1 (0.59) CYP1A2CYP2D6GABRA1GABRB2TSHR
SCHEMBL11803468 0.72 GABRA1 (0.59) CYP1A2CYP2D6GABRA1GABRB2FABP3
SCHEMBL14705354 0.71 GABRA1 (0.57) CYP1A2CYP2D6GABRA1GABRB2TSHR
SCHEMBL14703867 0.71 GABRA1 (0.57) CYP1A2CYP2D6GABRA1GABRB2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5106975-A Hexahydropyrimidine derivatives ETHYL PETROLEUM ADDITIVES, INC. (US) 1992-04-21 US disclosed
EP-0434185-A2 Hexahydropyrimidine derivatives ETHYL PETROLEUM ADDITIVES, INC. (US) 1991-06-26 EP disclosed