SCHEMBL9734334

SCHEMBL9734334

O=C(O)C1CN(c2ccccc2)C(=O)C1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
POLB P06746 3/20 0.41
NOTUM Q6P988 1/20 0.41
MAPT P10636 2/20 0.40
ALDH1A1 P00352 2/20 0.39
USP2 O75604 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GRM2 Q14416 1/20 0.37
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA4 P22748 2/20 0.37
CA6 P23280 2/20 0.37
CA7 P43166 2/20 0.37
CA9 Q16790 2/20 0.37
CA5B Q9Y2D0 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31530864 0.85 NOTUM (0.45) NPC1RAB9AKMT2AMEN1POLB
SCHEMBL7414405 0.74 KCNH2 (0.39) KMT2AMEN1ALDH1A1HPGDSMN1; SMN2
SCHEMBL308869 0.71 PTPN1 (0.59) NPC1RAB9AKMT2AMEN1POLB
SCHEMBL9043612 0.71 POLB (0.46) KMT2APOLBALDH1A1HPGDSMN1; SMN2
SCHEMBL9203728 0.70 NPC1 (0.46) NPC1RAB9AKMT2AMEN1MAPT
SCHEMBL9042425 0.69 GAA (0.41) KMT2AMEN1POLBMAPTALDH1A1
SCHEMBL8431884 0.69 PTPN1 (0.50) NPC1RAB9AKMT2AMEN1POLB
SCHEMBL15319525 0.68 PTPN1 (0.49) NPC1RAB9AKMT2AMEN1POLB
SCHEMBL11066860 0.68 NPC1 (0.47) NPC1RAB9AKMT2AMEN1POLB
SCHEMBL20116495 0.68 CA12 (0.66) NPC1KMT2AMEN1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132424-A Anticholesterol, treatment of atherosclerosis THE UPJOHN COMPANY (US) 1992-07-21 US disclosed
EP-0425541-A1 PYRAZOLO-AZOLO-PYRIMIDINE-DIONES THE UPJOHN COMPANY (US) 1991-05-08 EP disclosed
WO-1990001031-A1 PYRAZOLO-PYRROLO-PYRIMIDINE-DIONES THE UPJOHN COMPANY (US) 1990-02-08 WO disclosed