SCHEMBL308869

SCHEMBL308869

O=C(O)C1CCN(c2ccccc2)C1=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.59
USP30 Q70CQ3 1/20 0.53
ROCK2 O75116 2/20 0.50
ROCK1 Q13464 1/20 0.50
HDAC8 Q9BY41 3/20 0.48
HDAC6 Q9UBN7 3/20 0.48
HDAC1 Q13547 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
FPR1 P21462 1/20 0.47
FPR2 P25090 1/20 0.47
DDB1 Q16531 2/20 0.47
CRBN Q96SW2 2/20 0.47
NOTUM Q6P988 1/20 0.45
HSD11B1 P28845 1/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8431884 0.90 PTPN1 (0.50) PTPN1USP30ROCK2ROCK1HDAC8
SCHEMBL15319525 0.88 PTPN1 (0.49) PTPN1USP30ROCK2ROCK1HDAC8
SCHEMBL15374430 0.86 USP30 (0.51) PTPN1USP30ROCK2ROCK1HDAC8
SCHEMBL14943747 0.86 USP30 (0.51) PTPN1USP30ROCK2ROCK1HDAC8
SCHEMBL5104476 0.86 USP30 (0.51) PTPN1USP30ROCK2ROCK1HDAC8
SCHEMBL892180 0.85 PTPN1 (0.52) PTPN1USP30ROCK2ROCK1HDAC8
SCHEMBL1137236 0.85 PTPN1 (0.52) PTPN1USP30ROCK2MEN1KMT2A
SCHEMBL892417 0.85 HTT (0.54) PTPN1USP30ROCK2ROCK1MEN1
SCHEMBL6936690 0.85 PTPN1 (0.52) PTPN1USP30ROCK2ROCK1HDAC8
SCHEMBL892936 0.84 NOTUM (0.52) PTPN1USP30HDAC8HDAC6HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 131 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250346575-A1 ISOINDOLINONE DERIVATIVE HAVING GLUTARIMIDE MOTHER NUCLEUS, AND USE THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2025-11-13 US disclosed
US-20250276976-A1 CARDIAC SARCOMERE INHIBITORS CYTOKINETICS, INC. 2025-09-04 US disclosed
US-12275741-B2 Cardiac sarcomere inhibitors CYTOKINETICS, INC. (US) 2025-04-15 US disclosed
EP-4482832-A1 5-[7-(3,4-DIHYDRO-1H-ISOQUINOLINE-2-CARBONYL)-1,2,3,4 TETRAHYDROISOQUINOLIN-6-Y L]-1H-PYRROLE-3-CARBOXAMIDE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USES AS PRO-APOPTOTIC AGENTS Les Laboratoires Servier (FR) 2025-01-01 EP disclosed
CN-119053587-A 5- [7- (3, 4-Dihydro-1H-isoquinoline-2-carbonyl) -1,2,3,4 tetrahydroisoquinolin-6-yl ] -1H-pyrrole-3-carboxamide derivatives, pharmaceutical compositions containing same and use thereof as pro-apoptotic agents 法国施维雅药厂 2024-11-29 CN disclosed
CN-118955409-A Cardiac sarcomere inhibitors 赛特凯恩蒂克公司 2024-11-15 CN disclosed
US-20240368172-A1 CARDIAC SARCOMERE INHIBITORS CYTOKINETICS, INC. 2024-11-07 US disclosed
EP-4431505-A1 ISOINDOLINONE DERIVATIVE HAVING GLUTARIMIDE MOTHER NUCLEUS, AND USE THEREOF Korea Research Institute of Chemical Technology (KR) 2024-09-18 EP disclosed
CN-112867539-B Cardiac sarcomere inhibitors 赛特凯恩蒂克公司 2024-08-06 CN disclosed
CN-118234721-A Isoindolinone derivative with glutarimide mother nucleus and application thereof 韩国化学研究院 2024-06-21 CN disclosed
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE, INC. 2007-01-04 US disclosed
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE, INC. 2007-01-04 US disclosed
US-20030171578-A1 Pyrrolidinone derivative compound SCHERING AKTIENGESELLSCHAFT (DE) 2003-09-11 US disclosed
EP-0916656-B1 A method for production of pyrrolidinone derivatives SCHERING AG (DE) 2003-09-10 EP disclosed
US-6555694-B1 Reacting an aniline and cyclopropane-1,1-dicarboxylic acid; free of hydrogen-generating substance and moisture sensitive reagent; corrosion resistance; simplification; for piperazine derivatives used as central nervous system disorders SCHERING AKTIENGESELLSCHAFT (DE) 2003-04-29 US disclosed
US-6207825-B1 REACTING THE CORRESPONDING 3-CARBOXYPYRROLIDINONE COMPOUND IN THE PRESENCE OF FORMALDEHYDE MITSUI CHEMICALS, INC. (JP) 2001-03-27 US disclosed
JP-2000143624-A 3-CARBOXY-1-PHENYL-2-PYRROLIDINONE DERIVATIVE AND ITS PRODUCTION MITSUI CHEMICALS INC 2000-05-26 JP disclosed
EP-0916656-A2 A method for production of pyrrolidinone derivatives Mitsui Chemicals, Inc. (JP) 1999-05-19 EP disclosed
CN-1095066-A Weedicide ZENECA LTD (GB) 1994-11-16 CN disclosed
US-3970500-A PRESSURE SENSITIVE, FORMALDEHYDE-NAPHTHALENESULFONIC ACID FUJI PHOTO FILM CO., LTD. (JA) 1976-07-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling HGF, MET, FLT1 PTPN1 911/4885USP30 3430/4885ROCK2 242/4885
US-12275741-B2 Cardiac sarcomere inhibitors TNNI3, MYLK2, TNNT2 PTPN1 2251/4885USP30 2796/4885ROCK2 168/4885
US-20240368172-A1 CARDIAC SARCOMERE INHIBITORS TNNI3, MYLK2, TNNT2 PTPN1 2251/4885USP30 2796/4885ROCK2 168/4885
US-20250276976-A1 CARDIAC SARCOMERE INHIBITORS TNNI3, MYLK2, TNNT2 PTPN1 2251/4885USP30 2796/4885ROCK2 168/4885
US-20030171578-A1 Pyrrolidinone derivative compound PFAS, CBR1, PYCR1 PTPN1 1391/4885USP30 3214/4885ROCK2 2834/4885
US-20250346575-A1 ISOINDOLINONE DERIVATIVE HAVING GLUTARIMIDE MOTHER NUCLEUS, AND USE THEREOF CRBN, IDH1, IDH2 PTPN1 1412/4885USP30 2457/4885ROCK2 4396/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.