SCHEMBL9734960

SCHEMBL9734960

CC1(CO)C=C(n2ccccc2=O)c2cc(C#N)ccc2O1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 5/20 0.36
HTR1A P08908 4/20 0.34
ABCB1 P08183 5/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
MAOB P27338 1/20 0.33
F10 P00742 1/20 0.33
HTR2A P28223 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085392 0.91 HTR1A (0.35) ABCC9HTR1AABCB1PDE4APDE4B
SCHEMBL9735036 0.90 HTR1A (0.34) ABCC9HTR1AABCB1PDE4APDE4B
SCHEMBL9194883 0.88 PDE4A (0.36) ABCC9HTR1AABCB1PDE4APDE4B
Bimakalim SCHEMBL231904 0.86 PDE4A (0.43) ABCC9HTR1AABCB1PDE4APDE4B
SCHEMBL8088666 0.83 CASP3 (0.34) ABCC9HTR1AABCB1PDE4APDE4B
SCHEMBL9735833 0.81 CYP3A4 (0.38) ABCB1MAOB
SCHEMBL8133760 0.81 HTR1A (0.33) ABCC9HTR1APDE4APDE4BPDE4C
SCHEMBL8084380 0.79 OPRD1 (0.39) ABCC9HTR1APDE4APDE4BPDE4C
SCHEMBL8175110 0.79 OPRD1 (0.39) ABCC9HTR1APDE4APDE4BPDE4C
SCHEMBL8084291 0.78 OPRD1 (0.39) ABCC9HTR1APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5130322-A CHROMAN DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-14 US disclosed