SCHEMBL9735495

SCHEMBL9735495

CCc1cc(C(=O)CCCCC(=O)O)c(O)cc1OCCCCC#N

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 5/20 0.48
PDE5A O76074 6/20 0.45
PDE1A P54750 2/20 0.42
PDE1B Q01064 2/20 0.42
PDE1C Q14123 2/20 0.42
LTB4R Q15722 10/20 0.42
LTB4R2 Q9NPC1 5/20 0.41
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP3A4 P08684 1/20 0.38
THRB P10828 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
HTR2B P41595 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
SIGMAR1 Q99720 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9417917 0.99 NR1H4 (0.47) NR1H4PDE5APDE1APDE1BPDE1C
SCHEMBL9417949 0.87 PPARA (0.42) NR1H4PDE5AALDH1A1TSHR
SCHEMBL9417757 0.83 LTB4R (0.53) NR1H4PDE5ALTB4RLTB4R2MEN1
SCHEMBL9417971 0.82 LTB4R (0.53) NR1H4PDE5ALTB4RLTB4R2MEN1
SCHEMBL9417832 0.82 NR1H4 (0.49) NR1H4ALDH1A1THRBHPGD
SCHEMBL9735490 0.81 TSHR (0.37) LTB4RLTB4R2TSHR
SCHEMBL9417958 0.80 NR1H4 (0.56) NR1H4PDE5ALTB4RLTB4R2ALDH1A1
SCHEMBL9417862 0.79 PDE5A (0.60) NR1H4PDE5APDE1APDE1BPDE1C
SCHEMBL9417905 0.79 NR1H4 (0.48) NR1H4LTB4RLTB4R2ALDH1A1HPGD
SCHEMBL9417940 0.78 LTB4R (0.51) NR1H4LTB4RLTB4R2MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098613-A Aromatic ethers for treatment of mammals ELI LILLY AND COMPANY (US) 1992-03-24 US disclosed
US-4945099-A LEUKOTRIENE ANTAGONIST ELI LILLY AND COMPANY (US) 1990-07-31 US disclosed
EP-0276065-B1 ANTI-INFLAMMATORY AGENTS ELI LILLY AND COMPANY (US) 1990-06-06 EP disclosed
EP-0276065-A1 Anti-inflammatory agents ELI LILLY AND COMPANY (US) 1988-07-27 EP disclosed