SCHEMBL9735728

SCHEMBL9735728

COCC1(C)Cc2ccc(C#N)cc2C(OC2CCC(=O)C2)O1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 2/20 0.33
BACE1 P56817 11/20 0.33
ABCC9 O60706 2/20 0.32
ABCC8 Q09428 2/20 0.32
KCNJ11 Q14654 2/20 0.32
KCNJ8 Q15842 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
LMNA P02545 1/20 0.32
KCNH2 Q12809 1/20 0.32
ABCB1 P08183 1/20 0.32
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
DRD2 P14416 1/20 0.31
DRD3 P35462 1/20 0.31
CHRM2 P08172 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9735574 0.86 BACE1 (0.32) CYP11B2BACE1
SCHEMBL9737011 0.83 PNMT (0.34) DRD2
SCHEMBL9736993 0.74 ABCC9 (0.42) ABCC9ABCC8KCNJ11KCNJ8CYP1A2
SCHEMBL9735600 0.72 ABCC9 (0.51) BACE1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9197783 0.72 ABCB1 (0.34) BACE1ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9735704 0.72 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8CYP1A2
SCHEMBL9736523 0.66 SLC6A4 (0.39) CYP2D6CYP2C9CYP2C19KCNH2DRD3
SCHEMBL9198669 0.61 MAOB (0.44) ABCB1PDE4APDE4BPDE4CPDE4D
SCHEMBL9198396 0.60 ABCC9 (0.39) ABCC9ABCC8KCNJ11KCNJ8CYP1A2
SCHEMBL9735028 0.60 ABCC9 (0.37) BACE1ABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5130322-A CHROMAN DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-14 US disclosed
EP-0415065-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1991-03-06 EP disclosed