SCHEMBL9735949

SCHEMBL9735949

O=C1CCn2c1cc1cc(Cl)ccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
AHR P35869 1/20 0.36
VHL P40337 1/20 0.36
ELOC Q15369 1/20 0.36
ELOB Q15370 1/20 0.36
DRD3 P35462 1/20 0.36
SRD5A1 P18405 1/20 0.35
THRB P10828 2/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ACLY P53396 3/20 0.34
PTGS2 P35354 1/20 0.34
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844695 0.81 SIGMAR1 (0.39) THRBTP53KDM4EALDH1A1LMNA
SCHEMBL9259274 0.80 KDM4E (0.39) SRD5A1MAPTKDM4EALDH1A1LMNA
SCHEMBL946353 0.80 MEN1 (0.39) SRD5A1MAPTKDM4EALDH1A1LMNA
SCHEMBL9259549 0.77 HTR2A (0.44) HTR2AHTR2CDRD3KMT2A
SCHEMBL9736283 0.76 SRD5A1 (0.40) SRD5A1THRBMAPTKDM4EALDH1A1
SCHEMBL9264795 0.76 KDM4E (0.56) HTR2AHTR2CSRD5A1MAPTKDM4E
SCHEMBL30684298 0.72 ALOX5 (0.34)
SCHEMBL18850958 0.71 HTR2A (0.47) HTR2AHTR2C
SCHEMBL20777902 0.69 HTR2A (0.38) HTR2AHTR2CDRD3THRBTP53
SCHEMBL17907930 0.69 HTR2A (0.48) HTR2AHTR2CVHLELOCELOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992021678-A1 LIPOXYGENASE INHIBITING PYRROLO [1,2a]INDOLE COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1992-12-10 WO disclosed