SCHEMBL9735969

SCHEMBL9735969

O=C(O)C1(C(=O)c2ccccc2)CCc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC9 Q9UKV0 1/20 0.44
HCAR2 Q8TDS4 1/20 0.42
TDP1 Q9NUW8 2/20 0.39
LMNA P02545 1/20 0.39
KDM1A O60341 1/20 0.38
MAOB P27338 1/20 0.38
TSHR P16473 1/20 0.37
AKR1C1 Q04828 1/20 0.37
PIN1 Q13526 3/20 0.36
RBP4 P02753 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL433287 0.88 HDAC9 (0.50) HDAC9HCAR2TDP1KDM1AMAOB
Biphenyl SCHEMBL27506403 0.83 HDAC9 (0.46) HDAC9HCAR2TDP1KDM1AMAOB
Trimethylammonium SCHEMBL27680853 0.81 HDAC9 (0.45) HDAC9HCAR2TDP1LMNAKDM1A
SCHEMBL30219063 0.77 AKR1C1 (0.48) HDAC9HCAR2KDM1ATSHRAKR1C1
SCHEMBL687495 0.77 AKR1C1 (0.48) HDAC9HCAR2KDM1ATSHRAKR1C1
SCHEMBL27989169 0.75 SIGMAR1 (0.45) LMNAMAOB
SCHEMBL17335394 0.75 KDM1A (0.46) HDAC9HCAR2TDP1KDM1AMAOB
SCHEMBL7434294 0.74 SMN1; SMN2 (0.48) HDAC9LMNA
SCHEMBL5204567 0.74 HDAC9 (0.40) HDAC9HCAR2TDP1LMNAKDM1A
SCHEMBL31536279 0.73 HDAC9 (0.41) HDAC9HCAR2TDP1LMNAKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135940-A Antiallegens, antiinflammatory agents MERCK FROSST CANADA, INC. (CA) 1992-08-04 US disclosed
EP-0252639-A1 Leukotriene antagonists MERCK FROSST CANADA INC. (CA) 1988-01-13 EP disclosed