SCHEMBL9736677

SCHEMBL9736677

CC(=O)c1ccnc(CO)c1N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
PKM P14618 1/20 0.35
RAB9A P51151 1/20 0.35
KDM4E B2RXH2 3/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
KDM4C Q9H3R0 2/20 0.33
KDM5A P29375 1/20 0.33
KDM5B Q9UGL1 1/20 0.33
PRKCI P41743 1/20 0.33
LMNA P02545 1/20 0.32
GABRP O00591 1/20 0.32
GABRD O14764 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30345359 0.79 KDM4E (0.41) ALDH1A1L3MBTL1PDE3BPDE3AKMT2A
SCHEMBL25211812 0.79 KDM4E (0.41) ALDH1A1L3MBTL1PDE3BPDE3AKMT2A
SCHEMBL30898769 0.77 NOS3 (0.48) ALDH1A1SMN1; SMN2KDM4CPRKCI
SCHEMBL30590435 0.76 SMN1; SMN2 (0.42) ALDH1A1KMT2ASMN1; SMN2TP53KDM4E
SCHEMBL17619241 0.74 LMNA (0.40) ALDH1A1L3MBTL1KMT2ASMN1; SMN2KDM4E
SCHEMBL29472130 0.74 LMNA (0.40) ALDH1A1L3MBTL1KMT2ASMN1; SMN2KDM4E
SCHEMBL8534431 0.74 ALDH1A1 (0.57) ALDH1A1L3MBTL1SMN1; SMN2PKMKDM4E
SCHEMBL31277349 0.74 ALDH1A1 (0.57) ALDH1A1L3MBTL1SMN1; SMN2PKMKDM4E
SCHEMBL21198627 0.73 KDM4E (0.38) ALDH1A1L3MBTL1PDE3BPDE3AKDM4E
SCHEMBL17619234 0.71 KDM4E (0.37) ALDH1A1L3MBTL1PDE3BPDE3AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084458-A Bactericides, malaria and antitumor agents SCHAPER KLAUS JUERGEN (DE) 1992-01-28 US disclosed
EP-0200777-A1 NEW AMINO COMPOUNDS, PREPARATION PROCESS THEREOF, UTILIZATION THEREOF AND DRUGS CONTAINING THEM Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1986-11-12 EP disclosed
WO-1986002645-A1 NEW AMINO COMPOUNDS, PREPARATION PROCESS THEREOF, UTILIZATION THEREOF AND DRUGS CONTAINING THEM BYK GULDEN LOMBERG CHEMISCHE FABRIK GESELLSCHAFT M (DE) 1986-05-09 WO disclosed