SCHEMBL9737152

SCHEMBL9737152

CC1(C(=O)OCc2ccccc2)Oc2ccc(C#N)cc2C(=O)C1CN

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.46
ALOX15 P16050 1/20 0.46
ABCB1 P08183 10/20 0.39
ABCC9 O60706 1/20 0.35
GAA P10253 1/20 0.35
PKM P14618 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PTGER1 P34995 1/20 0.35
MAOB P27338 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9216559 0.71 CYP3A4 (0.54) CYP3A4ALOX15ABCB1ABCC9
SCHEMBL9737142 0.70 MAOB (0.42) CYP3A4ALOX15ABCB1GAAL3MBTL1
SCHEMBL9523872 0.67 TDP1 (0.43) CYP3A4ALOX15ABCB1ABCC9ALDH1A1
SCHEMBL9397793 0.65 CYP3A4 (0.81) CYP3A4ALOX15ABCB1
SCHEMBL9216547 0.65 CYP3A4 (0.58) CYP3A4ALOX15ABCB1ABCC9
SCHEMBL9216538 0.65 CYP3A4 (0.58) CYP3A4ALOX15ABCB1ABCC9
SCHEMBL9216552 0.65 CYP3A4 (0.58) CYP3A4ALOX15ABCB1ABCC9
SCHEMBL13790822 0.65 ALDH1A1 (0.49) L3MBTL1ALDH1A1
SCHEMBL10591175 0.64 CYP3A4 (0.80) CYP3A4ALOX15ABCB1
SCHEMBL9398521 0.64 CYP3A4 (0.80) CYP3A4ALOX15ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5130322-A CHROMAN DERIVATIVES MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-14 US disclosed
EP-0415065-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1991-03-06 EP disclosed