SCHEMBL9523872

SCHEMBL9523872

CC1(C)C=C(c2ccc(C(=O)OCc3ccccc3)cn2)c2cc(C#N)ccc2O1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.43
CYP3A4 P08684 1/20 0.40
ALOX15 P16050 1/20 0.40
LMNA P02545 3/20 0.38
KMT2A Q03164 2/20 0.38
CYP2D6 P10635 1/20 0.38
OPRD1 P41143 1/20 0.38
KCNH2 Q12809 1/20 0.38
TSHR P16473 1/20 0.37
ALDH1A1 P00352 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
JMJD6 Q6NYC1 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A3 Q01959 1/20 0.36
ABCC9 O60706 1/20 0.35
HIF1A Q16665 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9523558 0.85 RARA (0.42) KMT2ACYP2D6OPRD1KCNH2ABCC9
SCHEMBL9528002 0.79 KDM1A (0.36) KCNH2MAPTKDM4EABCC9ABCB1
SCHEMBL9525005 0.78 GABRA1 (0.38) OPRD1ABCC9
SCHEMBL9524497 0.76 GRM5 (0.39) ALDH1A1ABCC9ABCB1
SCHEMBL9628243 0.75 PDE4A (0.34) ABCC9ABCB1
SCHEMBL9525564 0.75 KDM1A (0.36) ABCC9ABCB1
SCHEMBL9524637 0.75 GRM5 (0.39) ABCC9
SCHEMBL8332841 0.74 METAP2 (0.40) KMT2ATSHRALDH1A1MAPTKDM4E
SCHEMBL9527814 0.74 PDE4A (0.34) ABCC9
Hydrochloric Acid SCHEMBL9627192 0.73 PDE4A (0.34) ABCC9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0298452-B1 2H-1-BENZOPYRANE DERIVATIVES SUBSTITUTED IN POSITION 4 BY ARYL OR N-HETEROARYL F. HOFFMANN-LA ROCHE AG (CH) 1993-06-30 EP disclosed
US-5118694-A Hypotensive agents; treatment for cardiovascular and muscular disorders HOFFMANN-LA ROCHE INC. (US) 1992-06-02 US disclosed
US-4971982-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS, SMOOTH MUSCLE DISORDERS HOFFMANN-LA ROCHE INC. (US) 1990-11-20 US disclosed
EP-0298452-A2 2H-1-benzopyrane derivatives substituted in position 4 by aryl or N-heteroaryl F. HOFFMANN-LA ROCHE AG (CH) 1989-01-11 EP disclosed