SCHEMBL9737978

SCHEMBL9737978

CC(C)NC(=O)c1nc(Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n(C(C)C)n1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 2/20 0.34
AGTR2 P50052 1/20 0.34
TSHR P16473 1/20 0.33
PTGS2 P35354 1/20 0.33
FAAH O00519 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MGLL Q99685 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9738134 0.93 AGTR1 (0.35) AGTR1AGTR2FAAHALDH1A1MGLL
SCHEMBL9738129 0.90 AGTR1 (0.35) AGTR1AGTR2
SCHEMBL9739512 0.90 AGTR1 (0.33) AGTR1AGTR2FAAHALDH1A1MGLL
SCHEMBL9738516 0.89 AGTR1 (0.36) AGTR1AGTR2
SCHEMBL9738653 0.88 TRPV1 (0.35) PTGS2ALDH1A1
SCHEMBL9738503 0.88 TRPV1 (0.36) TSHRPTGS2ALDH1A1
SCHEMBL9738276 0.87 AGTR1 (0.38) AGTR1AGTR2
SCHEMBL9738315 0.87 AGTR1 (0.41) AGTR1
SCHEMBL9738918 0.86 SLC33A1 (0.34) AGTR1
SCHEMBL9738630 0.85 AGTR1 (0.47) AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992005161-A1 1,3,5-TRISUBSTITUTED-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CIRCULATORY DISORDERS G.D. SEARLE & CO. (US) 1992-04-02 WO claimed
WO-1992005161-A1 1,3,5-TRISUBSTITUTED-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CIRCULATORY DISORDERS G.D. SEARLE & CO. (US) 1992-04-02 WO disclosed