SCHEMBL9738516

SCHEMBL9738516

CCCNC(=O)c1nc(Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n(C(C)C)n1

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 8/20 0.36
AGTR2 P50052 1/20 0.36
BRD4 O60885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9738276 0.95 AGTR1 (0.38) AGTR1AGTR2
SCHEMBL9738129 0.93 AGTR1 (0.35) AGTR1AGTR2
SCHEMBL9738134 0.90 AGTR1 (0.35) AGTR1AGTR2
SCHEMBL9737978 0.89 AGTR1 (0.34) AGTR1AGTR2
SCHEMBL9738567 0.87 AGTR1 (0.41) AGTR1
SCHEMBL9739512 0.87 AGTR1 (0.33) AGTR1AGTR2
SCHEMBL9738438 0.86 AGTR1 (0.36) AGTR1
SCHEMBL9738653 0.86 TRPV1 (0.35)
SCHEMBL9739973 0.86 AGTR1 (0.47) AGTR1
SCHEMBL9738503 0.85 TRPV1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992005161-A1 1,3,5-TRISUBSTITUTED-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CIRCULATORY DISORDERS G.D. SEARLE & CO. (US) 1992-04-02 WO claimed
WO-1992005161-A1 1,3,5-TRISUBSTITUTED-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CIRCULATORY DISORDERS G.D. SEARLE & CO. (US) 1992-04-02 WO disclosed