SCHEMBL9739512

SCHEMBL9739512

CC(C)n1nc(C(=O)Nc2ccccc2)nc1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 3/20 0.33
EDNRA P25101 1/20 0.33
FAAH O00519 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MGLL Q99685 1/20 0.33
BCHE P06276 1/20 0.33
CNR2 P34972 1/20 0.33
AGTR2 P50052 2/20 0.33
DGAT1 O75907 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9738134 0.91 AGTR1 (0.35) AGTR1FAAHALDH1A1MGLLAGTR2
SCHEMBL9737978 0.90 AGTR1 (0.34) AGTR1FAAHALDH1A1MGLLAGTR2
SCHEMBL9738129 0.89 AGTR1 (0.35) AGTR1AGTR2
SCHEMBL9738516 0.87 AGTR1 (0.36) AGTR1AGTR2
SCHEMBL9738276 0.86 AGTR1 (0.38) AGTR1AGTR2
SCHEMBL9738035 0.85 AGTR1 (0.41) AGTR1
SCHEMBL9738653 0.85 TRPV1 (0.35) ALDH1A1
SCHEMBL9738272 0.85 AGTR1 (0.35) AGTR1EDNRAAGTR2
SCHEMBL9738616 0.85 SLC33A1 (0.36) AGTR1EDNRAAGTR2
SCHEMBL9738503 0.84 TRPV1 (0.36) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992005161-A1 1,3,5-TRISUBSTITUTED-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CIRCULATORY DISORDERS G.D. SEARLE & CO. (US) 1992-04-02 WO claimed
WO-1992005161-A1 1,3,5-TRISUBSTITUTED-1,2,4-TRIAZOLE COMPOUNDS FOR TREATMENT OF CIRCULATORY DISORDERS G.D. SEARLE & CO. (US) 1992-04-02 WO disclosed