SCHEMBL9738560

SCHEMBL9738560

N#CC1(C#N)OC1c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.38
HPGD P15428 8/20 0.38
KMT2A Q03164 7/20 0.38
KDM4E B2RXH2 6/20 0.38
GLA P06280 5/20 0.38
GAA P10253 4/20 0.38
MEN1 O00255 5/20 0.37
THRB P10828 1/20 0.37
RECQL P46063 1/20 0.37
MAPT P10636 4/20 0.36
CASP1 P29466 2/20 0.34
CASP7 P55210 2/20 0.34
HSD17B10 Q99714 2/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
YWHAG P61981 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
TSHR P16473 2/20 0.33
KDM1A O60341 2/20 0.33
CUL4A Q13619 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10703931 0.81 MAPT (0.42) ALDH1A1KMT2AKDM4EGAAMEN1
SCHEMBL8178191 0.79 MAOB (0.55) GAAMAPTL3MBTL1CYP2C19LMNA
SCHEMBL6499286 0.77 DRD3 (0.43) CASP1TSHRKDM1A
SCHEMBL8173176 0.75 MAOB (0.47) KDM1A
SCHEMBL9059555 0.69 CHRNB2 (0.36) ALDH1A1HPGDKMT2AMEN1
SCHEMBL13318482 0.67 TSHR (0.39) ALDH1A1KMT2AKDM4EMEN1MAPT
SCHEMBL3972334 0.67 KDM1A (0.43) ALDH1A1KMT2AMEN1L3MBTL1TSHR
SCHEMBL17660056 0.67 KDM1A (0.43) ALDH1A1KMT2AMEN1L3MBTL1TSHR
SCHEMBL5955814 0.67 KDM1A (0.43) ALDH1A1KMT2AMEN1L3MBTL1TSHR
SCHEMBL18298261 0.67 TSHR (0.39) ALDH1A1KMT2AKDM4EMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116239573-B Preparation method and application of metal organic quaternary cyclic compound 大连理工大学 2024-03-26 CN disclosed
CN-116239573-A Preparation method and application of metal organic quaternary cyclic compound 大连理工大学 2023-06-09 CN disclosed
US-5082842-A Sedatives HOFFMANN-LA ROCHE INC. (US) 1992-01-21 US disclosed
US-4889854-A MUSCLE RELAXANT, SEDATIVE-HYPNOTIC, ANXIOLYTIC AND-OR ANTICONVULSANT ACTIVITY HOFFMAN-LA ROCHE INC. (US) 1989-12-26 US disclosed
EP-0294599-A2 Tricyclic pyridone derivatives F. HOFFMANN-LA ROCHE AG (CH) 1988-12-14 EP disclosed