SCHEMBL9738928

SCHEMBL9738928

COc1cc2c(cc1OC)CC(=O)N(CC1CCCCN(CCCOc3cccc4c(OC)c(OC)ccc34)C1)CC2

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.42
HRH3 Q9Y5N1 7/20 0.41
HCN4 Q9Y3Q4 2/20 0.39
MAPT P10636 1/20 0.39
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
KMT2A Q03164 1/20 0.38
CHRM2 P08172 1/20 0.37
HTR1A P08908 1/20 0.37
SLC6A4 P31645 1/20 0.37
DRD3 P35462 1/20 0.37
KCNH2 Q12809 1/20 0.37
S1PR5 Q9H228 1/20 0.36
ADRA1B P35368 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9740634 0.95 HRH3 (0.41) ABCB1HRH3HCN4MAPTCYP3A4
SCHEMBL9742239 0.91 ADRA1B (0.45) ABCB1HRH3MEN1ALDH1A1CYP1A2
SCHEMBL9740162 0.89 HRH3 (0.49) ABCB1HRH3MEN1ALDH1A1CYP1A2
SCHEMBL9739322 0.87 HRH3 (0.42) ABCB1HRH3
Hydrochloric Acid SCHEMBL9741913 0.86 HRH3 (0.39) ABCB1HRH3MEN1ALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL9740876 0.84 HRH3 (0.47) ABCB1HRH3MEN1ALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL9739352 0.84 ADRA1B (0.39) ABCB1HRH3MEN1ALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL9740789 0.82 KDM4E (0.48) ABCB1HRH3CYP3A4ALOX15ALDH1A1
SCHEMBL9215853 0.82 HCN4 (0.35) HCN4MAPTCYP3A4ALOX15MEN1
SCHEMBL9740254 0.80 HRH3 (0.44) ABCB1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed