SCHEMBL9738952

SCHEMBL9738952

CN(C)c1ncc2ncn(Cc3ccccc3F)c2n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 6/20 0.47
PDE4B Q07343 6/20 0.47
PDE4C Q08493 6/20 0.47
PDE4D Q08499 6/20 0.47
PDE5A O76074 3/20 0.47
PDE1A P54750 3/20 0.47
PDE1B Q01064 3/20 0.47
PDE1C Q14123 3/20 0.47
PDE3B Q13370 2/20 0.47
PDE3A Q14432 2/20 0.47
ALDH1A1 P00352 9/20 0.46
HSD17B10 Q99714 9/20 0.46
CYP1A2 P05177 8/20 0.46
CASP7 P55210 8/20 0.46
TSHR P16473 7/20 0.46
CASP1 P29466 7/20 0.46
CYP2C9 P11712 6/20 0.46
CYP2D6 P10635 6/20 0.46
CYP2C19 P33261 5/20 0.46
CYP3A4 P08684 5/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9740503 0.86 ACP1 (0.44) ALDH1A1HSD17B10CYP1A2CASP7TSHR
SCHEMBL9739221 0.86 ALDH1A1 (0.46) ALDH1A1HSD17B10CYP1A2CASP7TSHR
SCHEMBL9738484 0.80 FGFR1 (0.49) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL9739048 0.80 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL9738442 0.80 PDE4A (0.56) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL9741263 0.79 ADORA2A (0.52) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL9739371 0.77 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL11014177 0.77 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DPDE5A
Dimethylamine SCHEMBL4532702 0.77 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DPDE5A
SCHEMBL23228189 0.76 CYP1A2 (0.50) ALDH1A1HSD17B10CYP1A2CASP7TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0363320-A2 Substituted 9H purine CIBA-GEIGY AG (CH) 1990-04-11 EP claimed
US-5110818-A Antiepileptic agents CIBA-GEIGY CORPORATION (US) 1992-05-05 US disclosed
EP-0363320-A2 Substituted 9H purine CIBA-GEIGY AG (CH) 1990-04-11 EP disclosed