SCHEMBL9739221

SCHEMBL9739221

CN(C)c1ncc2ncn(Cc3c(F)cccc3F)c2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.46
HSD17B10 Q99714 11/20 0.46
CASP1 P29466 10/20 0.46
CASP7 P55210 10/20 0.46
CYP1A2 P05177 9/20 0.46
TSHR P16473 8/20 0.46
CYP2C9 P11712 7/20 0.46
CYP3A4 P08684 7/20 0.46
CYP2C19 P33261 6/20 0.46
HPGD P15428 4/20 0.46
CYP2D6 P10635 4/20 0.46
USP2 O75604 5/20 0.45
CLK4 Q9HAZ1 2/20 0.45
HIF1A Q16665 5/20 0.42
MAPK1 P28482 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KCNH2 Q12809 1/20 0.42
LMNA P02545 1/20 0.41
ADORA2A P29274 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9738952 0.86 PDE4A (0.47) ALDH1A1HSD17B10CASP1CASP7CYP1A2
SCHEMBL9738831 0.80 FGFR1 (0.50) ALDH1A1TSHRMAPK1ADORA2AADORA1
SCHEMBL9738800 0.80 PDE4A (0.50) LMNAADORA2AADORA1AXLMERTK
SCHEMBL9738685 0.79 AXL (0.47) TSHRMAPK1ADORA2AADORA1AXL
SCHEMBL9739172 0.79 ADORA2A (0.51) ADORA2AADORA1AXLMERTKFLT3
SCHEMBL23228189 0.77 CYP1A2 (0.50) ALDH1A1HSD17B10CASP1CASP7CYP1A2
SCHEMBL9740503 0.77 ACP1 (0.44) ALDH1A1HSD17B10CASP1CASP7CYP1A2
SCHEMBL9740123 0.77 AXL (0.61) ADORA2AADORA1AXLMERTKFLT3
SCHEMBL23867154 0.76 CYP1A2 (0.49) ALDH1A1HSD17B10CASP1CASP7CYP1A2
SCHEMBL10442061 0.71 CYP1A2 (0.61) CYP1A2CYP2D6MAPK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110818-A Antiepileptic agents CIBA-GEIGY CORPORATION (US) 1992-05-05 US disclosed
EP-0363320-A2 Substituted 9H purine CIBA-GEIGY AG (CH) 1990-04-11 EP disclosed