SCHEMBL9739003

SCHEMBL9739003

CCCCc1nc(C)c(CC)c(Cl)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 3/20 0.36
TLR7 Q9NYK1 3/20 0.36
ALDH1A1 P00352 4/20 0.34
CETP P11597 1/20 0.34
RXFP1 Q9HBX9 2/20 0.33
HTT P42858 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
POLB P06746 1/20 0.33
KDM4E B2RXH2 1/20 0.33
TYMP P19971 1/20 0.33
PDE4A P27815 2/20 0.31
PDE4B Q07343 2/20 0.31
PDE4C Q08493 2/20 0.31
PDE4D Q08499 2/20 0.31
CYP1A2 P05177 2/20 0.31
CYP2C9 P11712 2/20 0.31
CYP2C19 P33261 2/20 0.31
CYP2D6 P10635 1/20 0.31
LMNA P02545 1/20 0.31
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9738686 0.81 PDE4A (0.33) TLR8TLR7ALDH1A1CETPTYMP
Acetic Acid SCHEMBL9257350 0.79 PDE4A (0.35) ALDH1A1RXFP1HTTPOLBPDE4A
SCHEMBL5158467 0.78 PDE10A (0.35) ALDH1A1CETPTYMPPDE4APDE4B
SCHEMBL9843662 0.78 MAPT (0.37) TLR8TLR7ALDH1A1RXFP1HTT
SCHEMBL9739507 0.78 TLR8 (0.42) TLR8TLR7
SCHEMBL649969 0.75 TLR8 (0.39) TLR8TLR7ALDH1A1HTTKDM4E
SCHEMBL855416 0.74 CYP1A2 (0.31) RXFP1CYP1A2CYP2C9CYP2C19CYP2D6
SCHEMBL13531385 0.74 TLR8 (0.43) TLR8TLR7ALDH1A1HTTSMN1; SMN2
SCHEMBL16229359 0.73 TYMP (0.34) TLR8TLR7ALDH1A1HTTSMN1; SMN2
SCHEMBL16229360 0.73 GCGR (0.36) TLR8TLR7ALDH1A1HTTTYMP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5100897-A Hypotensive agents, congestive heart failure, ocular hypertension MERCK & CO., INC. (US) 1992-03-31 US disclosed
EP-0419048-A2 Substituted pyrimidinones as angiotensin II antagonists MERCK & CO. INC. (US) 1991-03-27 EP disclosed