SCHEMBL5158467

SCHEMBL5158467

CCCCc1nc(Cl)c(C)c(Cl)n1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.35
PDE4A P27815 6/20 0.35
PDE4B Q07343 6/20 0.35
PDE4C Q08493 6/20 0.35
PDE4D Q08499 6/20 0.35
CETP P11597 1/20 0.35
PDE3B Q13370 4/20 0.33
PDE3A Q14432 4/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
ALDH1A1 P00352 2/20 0.33
SIRT1 Q96EB6 1/20 0.33
TYMP P19971 1/20 0.33
NOS2 P35228 1/20 0.33
PDK2 Q15119 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CASP1 P29466 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9738686 0.90 PDE4A (0.33) PDE10APDE4APDE4BPDE4CPDE4D
SCHEMBL9739003 0.78 TLR8 (0.36) PDE4APDE4BPDE4CPDE4DCETP
SCHEMBL12251371 0.77 CASP1 (0.41) PDE4APDE4BPDE4CPDE4DCETP
SCHEMBL1318651 0.76 ALDH1A1 (0.40) PDE4APDE4BPDE4CPDE4DCETP
SCHEMBL10911101 0.76 CETP (0.36) PDE4APDE4BPDE4CPDE4DCETP
SCHEMBL1187479 0.73 NOS2 (0.36) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL1321965 0.73 KMT2A (0.39) PDE4APDE4BPDE4CPDE4DCETP
SCHEMBL11679118 0.72 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL16229359 0.72 TYMP (0.34) PDE4APDE4BPDE4CPDE4DL3MBTL1
SCHEMBL16229360 0.72 GCGR (0.36) L3MBTL1ALDH1A1SIRT1TYMPNOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1747222-A1 PYRIMIDINE DERIVATIVES ANTAGONISTS OF VITRONECTIN RECEPTOR Proskelia SAS (FR) 2007-01-31 EP disclosed
WO-2005123734-A1 PYRIMIDINE DERIVATIVES ANTAGONISTS OF VITRONECTIN RECEPTOR PROSKELIA SAS (FR) 2005-12-29 WO disclosed