SCHEMBL9739386

SCHEMBL9739386

O=C1Cc2ccc3c(c2CCN1)OCO3

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 6/20 0.43
CYP2D6 P10635 5/20 0.43
CYP3A4 P08684 4/20 0.43
KDM4E B2RXH2 3/20 0.43
TSHR P16473 3/20 0.43
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
NQO2 P16083 2/20 0.36
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA7 P36544 1/20 0.34
CHRNA4 P43681 1/20 0.34
CYP1A2 P05177 3/20 0.33
TXNRD1 Q16881 1/20 0.33
TXNRD3 Q86VQ6 1/20 0.33
TXNRD2 Q9NNW7 1/20 0.33
ALDH1A1 P00352 1/20 0.33
XBP1 P17861 1/20 0.33
CYP19A1 P11511 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319733 0.79 CYP2D6 (0.46) CYP2C19CYP2D6CYP3A4KDM4ETSHR
SCHEMBL232442 0.77 HTR2C (0.44) CYP2C19CYP2D6CYP3A4KDM4ETSHR
SCHEMBL11336504 0.75 CYP2D6 (0.45) CYP2C19CYP2D6CYP3A4KDM4ETSHR
SCHEMBL9739665 0.73 KDM4E (0.60) CYP2C19CYP2D6KDM4ECHRNA7CYP1A2
SCHEMBL7478754 0.72 AHR (0.42) CYP2C19CYP2D6CYP3A4KDM4ETSHR
SCHEMBL4701400 0.71 GRIA2 (0.35) CYP2C19CYP2D6CYP3A4KDM4ETSHR
SCHEMBL3872994 0.69 PNMT (0.46) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL9835971 0.69 POLB (0.41) CYP2C19CYP2D6CYP3A4KDM4ETSHR
SCHEMBL14640411 0.68 CYP2D6 (0.62) CYP2C19CYP2D6CYP3A4KDM4ETSHR
SCHEMBL24265578 0.67 PARP10 (0.57) MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed