SCHEMBL9739670

SCHEMBL9739670

COc1ccc(CCN2CCC(CN3C=Cc4cc(OC)c(OC)cc4CC3=O)C2)cc1OC

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCN4 Q9Y3Q4 6/20 0.55
BRD4 O60885 1/20 0.46
HTR1A P08908 1/20 0.44
SLC6A4 P31645 1/20 0.44
ABCB1 P08183 1/20 0.43
MAPT P10636 1/20 0.41
HSP90AA1 P07900 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HTT P42858 1/20 0.41
DHCR7 Q9UBM7 1/20 0.41
CYP3A4 P08684 1/20 0.41
ALOX15 P16050 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9740380 0.95 HCN4 (0.54) HCN4BRD4MAPTHSP90AA1ALDH1A1
SCHEMBL9739668 0.95 HCN4 (0.54) HCN4BRD4MAPTHSP90AA1ALDH1A1
Hydrochloric Acid SCHEMBL10766227 0.94 HCN4 (0.53) HCN4BRD4MAPTCYP3A4ALOX15
Hydrochloric Acid SCHEMBL9738862 0.85 HCN4 (0.44) HCN4MAPTALDH1A1
SCHEMBL9212968 0.83 ACHE (0.48) HCN4BRD4
Hydrochloric Acid SCHEMBL9739487 0.82 ACHE (0.47) HCN4BRD4
SCHEMBL9215863 0.81 BRD4 (0.40) HCN4BRD4ABCB1
SCHEMBL9739280 0.80 HCN4 (0.59) HCN4HTR1ASLC6A4ABCB1MAPT
SCHEMBL10756420 0.80 HCN4 (0.38) HCN4HTR1ASLC6A4MAPTALDH1A1
SCHEMBL9740666 0.79 ABCB1 (0.41) HTR1ASLC6A4ABCB1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0224794-B1 CYCLIC AMINE DERIVATIVES, MEDICINES CONTAINING THESE COMPOUNDS AND PROCESS FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1990-09-12 EP disclosed
EP-0224794-A2 Cyclic amine derivatives, medicines containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1987-06-10 EP disclosed