SCHEMBL9740666

SCHEMBL9740666

CO/C1=C\C=C/N(CC2CCN(CCc3ccc(OC)c(OC)c3)C2)C(=O)Cc2ccccc2C1OC

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.41
SMPD1 P17405 1/20 0.40
HTR1A P08908 1/20 0.38
SLC6A4 P31645 1/20 0.38
EBP Q15125 2/20 0.38
SIGMAR1 Q99720 2/20 0.38
TMEM97 Q5BJF2 1/20 0.38
POLB P06746 1/20 0.37
MAPK1 P28482 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9739670 0.79 HCN4 (0.55) ABCB1HTR1ASLC6A4ALDH1A1
SCHEMBL9739668 0.74 HCN4 (0.54) SMPD1SIGMAR1ALDH1A1
SCHEMBL9740380 0.74 HCN4 (0.54) SMPD1SIGMAR1ALDH1A1
Hydrochloric Acid SCHEMBL10766227 0.73 HCN4 (0.53) SMPD1
SCHEMBL9739280 0.72 HCN4 (0.59) ABCB1SMPD1HTR1ASLC6A4MAPK1
SCHEMBL9740673 0.70 ABCB1 (0.43) ABCB1SMPD1HTR1ASLC6A4EBP
Hydrochloric Acid SCHEMBL9738862 0.69 HCN4 (0.44) ALDH1A1TSHRSMN1; SMN2
SCHEMBL9739025 0.68 HTR1A (0.56) ABCB1HTR1ASLC6A4EBPSIGMAR1
Cilobradine SCHEMBL1855245 0.68 HCN4 (0.57) SMPD1HTR1ASLC6A4SIGMAR1POLB
Cilobradine SCHEMBL30169956 0.68 HCN4 (0.57) SMPD1HTR1ASLC6A4SIGMAR1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed