SCHEMBL9739720

SCHEMBL9739720

COc1cc2c(cc1Cl)CCN(CC1CCCN(CCc3ccccc3)C1)C(=O)C2

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 2/20 0.47
CHRNB2 P17787 3/20 0.45
CHRNB4 P30926 3/20 0.45
CHRNA3 P32297 3/20 0.45
CHRNA4 P43681 3/20 0.45
KCNH2 Q12809 1/20 0.43
GAA P10253 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MAPT P10636 1/20 0.41
HCN4 Q9Y3Q4 1/20 0.41
CYP3A4 P08684 1/20 0.40
ALOX15 P16050 1/20 0.40
HTR1A P08908 1/20 0.39
SLC6A4 P31645 1/20 0.39
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9740561 0.94 CHRNB2 (0.49) CCR2CHRNB2CHRNB4CHRNA3CHRNA4
Hydrochloric Acid SCHEMBL9739064 0.93 CHRNB2 (0.48) CCR2CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9746442 0.91 CHRNB2 (0.46) CHRNB2CHRNB4CHRNA3CHRNA4GAA
SCHEMBL9740942 0.91 CCR2 (0.52) CCR2CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9742193 0.91 HCN4 (0.52) KCNH2GAAMEN1KMT2AMAPT
SCHEMBL9739855 0.91 CHRNB2 (0.46) CCR2CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9740796 0.90 CHRNB2 (0.45) CCR2CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9739409 0.90 CHRNB2 (0.47) CCR2CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9740124 0.87 HCN4 (0.51) GAAMEN1KMT2AMAPTHCN4
SCHEMBL9740542 0.86 GAA (0.42) CCR2CHRNB2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0224794-A2 Cyclic amine derivatives, medicines containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1987-06-10 EP disclosed