SCHEMBL9739898

SCHEMBL9739898

CN(C)c1nc(N)nc2c1ncn2Cc1ccccc1Cl

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.51
PDE4B Q07343 1/20 0.51
PDE4C Q08493 1/20 0.51
PDE4D Q08499 1/20 0.51
PDE3B Q13370 1/20 0.51
PDE3A Q14432 1/20 0.51
ADORA2A P29274 5/20 0.48
YTHDC1 Q96MU7 1/20 0.47
CNR2 P34972 4/20 0.46
ACP1 P24666 1/20 0.46
HSP90AA1 P07900 2/20 0.45
HSP90AB1 P08238 2/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
HIF1A Q16665 1/20 0.45
PHLPP2 Q6ZVD8 1/20 0.45
ADORA1 P30542 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9738569 0.88 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9739561 0.87 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9738116 0.86 ADORA2A (0.60) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9739040 0.84 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9738563 0.84 CDK1 (0.55) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9738222 0.82 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9739343 0.81 YTHDC1 (0.68) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9738722 0.81 ADORA2A (0.48) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9475371 0.79 CNR2 (0.51) ADORA2ACNR2ALDH1A1ADORA1
SCHEMBL27580729 0.77 CDK1 (0.46) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110818-A Antiepileptic agents CIBA-GEIGY CORPORATION (US) 1992-05-05 US disclosed
EP-0363320-A2 Substituted 9H purine CIBA-GEIGY AG (CH) 1990-04-11 EP disclosed