SCHEMBL9738563

SCHEMBL9738563

Nc1nc(N)c2ncn(Cc3ccccc3Cl)c2n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.55
CCNB1 P14635 1/20 0.55
CCNE1 P24864 1/20 0.55
CDK2 P24941 1/20 0.55
ADORA2A P29274 7/20 0.53
HSP90AA1 P07900 2/20 0.50
HSP90AB1 P08238 2/20 0.50
PDE4A P27815 1/20 0.50
PDE4B Q07343 1/20 0.50
PDE4C Q08493 1/20 0.50
PDE4D Q08499 1/20 0.50
ACP1 P24666 1/20 0.50
YTHDC1 Q96MU7 1/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
HIF1A Q16665 1/20 0.49
PHLPP2 Q6ZVD8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9738574 0.84 ADORA2A (0.66) CDK1CCNB1CCNE1CDK2ADORA2A
SCHEMBL9739343 0.84 YTHDC1 (0.68) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL9738444 0.84 YTHDC1 (0.56) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL9738722 0.84 ADORA2A (0.48) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL9739898 0.84 PDE4A (0.51) ADORA2AHSP90AA1HSP90AB1PDE4APDE4B
SCHEMBL1640041 0.83 PDE4A (0.69) CDK1CCNB1CCNE1CDK2ADORA2A
SCHEMBL11813045 0.82 ADORA2A (0.70) ADORA2AACP1ADORA1PI4KAPI4K2B
SCHEMBL9739774 0.82 ADORA2A (0.55) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL4358828 0.81 CDK1 (0.51) CDK1CCNB1CCNE1CDK2ADORA2A
SCHEMBL3273415 0.80 ADORA2A (0.78) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5110818-A Antiepileptic agents CIBA-GEIGY CORPORATION (US) 1992-05-05 US disclosed
EP-0363320-A2 Substituted 9H purine CIBA-GEIGY AG (CH) 1990-04-11 EP disclosed