SCHEMBL9740236

SCHEMBL9740236

CS(=O)(=O)c1ccc2c(c1)C(=O)Cc1ccccc1O2

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
BRD4 O60885 3/20 0.43
EPHX2 P34913 2/20 0.38
EPHX1 P07099 1/20 0.37
PTGS2 P35354 8/20 0.37
PTGS1 P23219 3/20 0.37
BCHE P06276 1/20 0.37
CES1 P23141 1/20 0.37
ACSL1 P33121 1/20 0.35
DRD3 P35462 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4427203 0.77 MAOA (0.61) MAOAMAOBBCHECES1
SCHEMBL5642473 0.77 MAOB (0.48) MAOAMAOBEPHX2BCHECES1
SCHEMBL10844098 0.77 AHR (0.49) MAOAMAOBBCHECES1ACSL1
SCHEMBL2375779 0.77 HPGD (0.52) MAOAMAOBDRD3
SCHEMBL9740773 0.76 MAOA (0.44) MAOAMAOBBRD4PTGS2PTGS1
SCHEMBL14598854 0.76 MAOA (0.44) MAOAMAOBPTGS2PTGS1BCHE
SCHEMBL19820969 0.76 MAOA (0.44) MAOAMAOBBCHECES1ACSL1
SCHEMBL10443908 0.74 PTGS2 (0.41) PTGS2PTGS1
SCHEMBL5658535 0.73 MAOA (0.52) MAOAMAOBBCHECES1ACSL1
SCHEMBL9493015 0.72 GAA (0.58) MAOAMAOBBRD4PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5140027-A Antidepressants, analgesics and anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-08-18 US disclosed
US-4943571-A ANALGESICS, ANTICONVULSANTS, ANTIDEPRESSANTS HOECHST-ROUSSEL PHAMRACEUTICALS INC. (US) 1990-07-24 US disclosed
US-4837227-A ANALGESICS, ANTIDEPRESSANTS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1989-06-06 US disclosed
EP-0002508-B1 AMINOALKYLTHIODIBENZOXEPINES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM HOECHST AKTIENGESELLSCHAFT (DE) 1982-03-31 EP disclosed