SCHEMBL9740673

SCHEMBL9740673

COC1=C(OC)c2ccccc2CC(=O)N(CC2CCN(CCc3ccc(OC)c(OC)c3)C2)CC=C1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.43
EBP Q15125 2/20 0.40
SIGMAR1 Q99720 2/20 0.40
TMEM97 Q5BJF2 1/20 0.40
MAPT P10636 1/20 0.40
HCN4 Q9Y3Q4 1/20 0.40
CYP3A4 P08684 1/20 0.40
ALOX15 P16050 1/20 0.40
SMPD1 P17405 1/20 0.39
HTR1A P08908 1/20 0.39
SLC6A4 P31645 1/20 0.39
POLB P06746 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9739280 0.78 HCN4 (0.59) ABCB1MAPTHCN4CYP3A4ALOX15
SCHEMBL9206607 0.74 ADRA1B (0.49) ABCB1MAPTHCN4CYP3A4ALOX15
Hydrochloric Acid SCHEMBL9213924 0.74 ADRA1B (0.49) ABCB1MAPTHCN4CYP3A4ALOX15
Cilobradine SCHEMBL628133 0.73 HCN4 (0.57) SIGMAR1MAPTHCN4CYP3A4ALOX15
Cilobradine SCHEMBL30169956 0.73 HCN4 (0.57) SIGMAR1MAPTHCN4CYP3A4ALOX15
Cilobradine SCHEMBL1855245 0.73 HCN4 (0.57) SIGMAR1MAPTHCN4CYP3A4ALOX15
Cilobradine SCHEMBL9518220 0.72 CYP3A4 (0.58) SIGMAR1MAPTHCN4CYP3A4ALOX15
SCHEMBL9215483 0.72 HTR1A (0.44) ABCB1MAPTHCN4CYP3A4ALOX15
Cilobradine SCHEMBL9740702 0.72 HCN4 (0.56) SIGMAR1MAPTHCN4CYP3A4ALOX15
Cilobradine SCHEMBL2459609 0.72 CYP3A4 (0.58) SIGMAR1MAPTHCN4CYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed