SCHEMBL9740950

SCHEMBL9740950

CCCc1cc(Cl)c2oc(-c3ccccc3)c(C)c2c1OC(C)=O

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 7/20 0.46
ADORA3 P0DMS8 2/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
BACE1 P56817 2/20 0.39
ALOX15 P16050 1/20 0.39
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
CREB1 P16220 1/20 0.35
PPARG P37231 1/20 0.35
PPARA Q07869 1/20 0.35
FPR1 P21462 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9739801 0.81 ALOX5 (0.67) ALOX5KDM4EALDH1A1ALOX15
SCHEMBL9740445 0.77 ALOX5 (0.64) ALOX5ALOX15FPR1
SCHEMBL9741057 0.77 ALOX5 (0.44) ALOX5KDM4EALDH1A1ALOX15PPARG
SCHEMBL9742551 0.76 ALOX5 (0.61) ALOX5ALOX15
SCHEMBL9739661 0.75 ALOX5 (0.72) ALOX5ALDH1A1ALOX15FPR1
SCHEMBL11022249 0.71 ALOX5 (0.35) ALOX5KDM4EALOX15PPARGPPARA
SCHEMBL9739794 0.71 ALOX5 (0.44) ALOX5KDM4EALDH1A1HPGDALOX15
SCHEMBL10738798 0.70 KDM4E (0.39) ALOX5ADORA3KDM4EALDH1A1HPGD
SCHEMBL9740742 0.69 ALOX5 (0.37) ALOX5ALOX15PPARGPPARA
SCHEMBL9739829 0.64 ALOX5 (0.60) ALOX5KDM4EALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5087638-A Inhibitors of mammalian leukotriene biosynthesis MERCK FROSST CANADA, INC. (CA) 1992-02-11 US disclosed
EP-0338782-A1 Benzofuran derivatives MERCK FROSST CANADA INC. (CA) 1989-10-25 EP disclosed
US-4863958-A TREATING ALLERGIC CONDITIONS, ASTHMA, CARDIOVASCULAR DISORDERS, AND INFLAMMATION MERCK FROSST CANADA, INC. (CA) 1989-09-05 US disclosed