SCHEMBL9743255

SCHEMBL9743255

O=C1c2ccc(Cl)cc2C2(c3ccc(F)cc3)CCCN12

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 5/20 0.40
ADAM17 P78536 2/20 0.38
ADAM10 O14672 1/20 0.38
MMP1 P03956 1/20 0.38
MMP2 P08253 1/20 0.38
MMP14 P50281 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MDM2 Q00987 3/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CNR1 P21554 2/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
AKR1B1 P15121 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9741939 0.92 SMN1; SMN2 (0.43) CHRM5HTTSMN1; SMN2MDM2CYP1A2
SCHEMBL9742447 0.90 ADAM17 (0.40) CHRM5ADAM17ADAM10MMP1MMP2
SCHEMBL9742194 0.88 SMN1; SMN2 (0.43) CHRM5HTTSMN1; SMN2MDM2CYP11B1
SCHEMBL9743860 0.87 HTT (0.41) CHRM5HTTSMN1; SMN2MDM2CYP1A2
SCHEMBL9743551 0.87 PSEN1 (0.40) CHRM5HTTSMN1; SMN2MDM2CYP1A2
SCHEMBL9743820 0.87 CHRM5 (0.45) CHRM5HTTSMN1; SMN2MDM2CYP1A2
SCHEMBL9743475 0.84 CHRM5 (0.45) CHRM5HTTSMN1; SMN2MDM2CYP2C9
SCHEMBL9742794 0.84 HTT (0.40) CHRM5HTTSMN1; SMN2CYP1A2CYP2D6
SCHEMBL9739646 0.82 CHRM5 (0.42) CHRM5AKR1B1
SCHEMBL9738615 0.82 CHRM5 (0.46) CHRM5HTTSMN1; SMN2MDM2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992016529-A1 NOVEL ISOINDOLE DERIVATIVES AND MEDICAMENTS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1992-10-01 WO disclosed