SCHEMBL9738615

SCHEMBL9738615

O=C1c2ccccc2C2(c3ccc(F)cc3)CCCN12

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 9/20 0.46
MAPT P10636 1/20 0.44
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41
PGR P06401 1/20 0.41
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
AKR1B1 P15121 1/20 0.39
MDM2 Q00987 2/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9739497 0.86 MAPT (0.46) CHRM5MAPTNPC1POLBPGR
SCHEMBL9739008 0.86 SMN1; SMN2 (0.55) CHRM5PGRHTTSMN1; SMN2MDM2
SCHEMBL9741164 0.85 CHRM5 (0.49) CHRM5NPC1POLBHTTSMN1; SMN2
SCHEMBL9739787 0.85 CHRM5 (0.43) CHRM5MAPTNPC1POLBPGR
SCHEMBL9740491 0.84 MEN1 (0.40) CHRM5MAPTNPC1POLBPGR
SCHEMBL9741279 0.84 PARK7 (0.43) CHRM5MAPTNPC1POLBMEN1
SCHEMBL9739646 0.84 CHRM5 (0.42) CHRM5MAPTNPC1POLBAKR1B1
SCHEMBL9738986 0.83 RXFP1 (0.42) CHRM5NPC1POLBHTTSMN1; SMN2
SCHEMBL9740223 0.83 CHRM5 (0.48) CHRM5MAPTNPC1PGRSMN1; SMN2
SCHEMBL9743255 0.82 CHRM5 (0.40) CHRM5HTTSMN1; SMN2AKR1B1MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992016529-A1 NOVEL ISOINDOLE DERIVATIVES AND MEDICAMENTS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1992-10-01 WO disclosed