SCHEMBL9745279

SCHEMBL9745279

CCOC(=O)C1=C(C=Cc2cc(CN(CC)CC)c(O)c(OC)c2)NC(C)=C(C(=O)OC)C1c1cccc(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 8/20 0.47
HIF1A Q16665 3/20 0.46
MEN1 O00255 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
KMT2A Q03164 2/20 0.46
MAPT P10636 2/20 0.46
LMNA P02545 1/20 0.46
POLB P06746 1/20 0.46
MAPK1 P28482 1/20 0.46
GPR55 Q9Y2T6 1/20 0.46
CYP2D6 P10635 1/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46
THPO P40225 1/20 0.46
ADORA3 P0DMS8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9745152 0.85 CACNA1B (0.51) CACNA1BHIF1AMEN1CYP1A2CYP3A4
SCHEMBL9745272 0.83 HIF1A (0.45) CACNA1BHIF1AMEN1CYP1A2CYP3A4
SCHEMBL9502243 0.76 ADORA3 (0.73) CACNA1BHIF1AMEN1CYP1A2CYP3A4
SCHEMBL10786311 0.75 CACNA1B (0.56) CACNA1BHIF1AMEN1CYP1A2CYP3A4
SCHEMBL9744641 0.74 CACNA1C (0.52) CACNA1BHIF1AMEN1CYP1A2CYP3A4
SCHEMBL9744636 0.74 CACNA1C (0.52) CACNA1BHIF1AMEN1CYP1A2CYP3A4
SCHEMBL3026966 0.72 ABCC1 (0.71) CACNA1BHIF1AMEN1CYP1A2CYP3A4
SCHEMBL9744740 0.72 CACNA1B (0.55) CACNA1BADORA3
SCHEMBL9744269 0.72 CACNA1C (0.65) CACNA1BHIF1AMEN1CYP1A2CYP3A4
SCHEMBL9744281 0.72 CACNA1C (0.65) CACNA1BHIF1AMEN1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0215250-B1 2-SUBSTITUTED-1,4-DIHYDROPYRIDINES, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1992-12-30 EP disclosed
US-4845113-A USEFUL IN RADICAL SCAVENGING THERAPY BOEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1989-07-04 US disclosed