SCHEMBL9745378

SCHEMBL9745378

CN1CCN(c2c(F)cc3c(=O)c(C(=O)OCC4=C(C(=O)O)N5C(=O)[C@@H](NC(=O)/C=N\OC(C(=O)O)c6csc(N)n6)[C@H]5SC4)cn(CCF)c3c2F)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
NR1I2 O75469 6/20 0.41
MAPT P10636 5/20 0.41
SLC22A6 Q4U2R8 3/20 0.41
SLC22A8 Q8TCC7 3/20 0.41
SLC22A11 Q9NSA0 3/20 0.41
PPARG P37231 2/20 0.41
ALB P02768 1/20 0.41
HTR2C P28335 1/20 0.39
TDP1 Q9NUW8 5/20 0.36
HPGD P15428 2/20 0.36
PGR P06401 2/20 0.35
DNMT1 P26358 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
L3MBTL1 Q9Y468 3/20 0.35
APEX1 P27695 2/20 0.35
ABCC4 O15439 2/20 0.35
CYP1A2 P05177 1/20 0.35
PKM P14618 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL9844206 0.88 KDM4E (0.42) KDM4ENR1I2MAPTSLC22A6SLC22A8
SCHEMBL30229691 0.83 NR1I2 (0.62) NR1I2MAPTSLC22A6SLC22A8SLC22A11
SCHEMBL9745004 0.83 NR1I2 (0.62) NR1I2MAPTSLC22A6SLC22A8SLC22A11
Hydrochloric Acid SCHEMBL9844164 0.83 NR1I2 (0.62) NR1I2MAPTSLC22A6SLC22A8SLC22A11
SCHEMBL9744140 0.82 KDM4E (0.56) KDM4ENR1I2MAPTSLC22A6SLC22A8
SCHEMBL9744130 0.82 KDM4E (0.56) KDM4ENR1I2MAPTSLC22A6SLC22A8
SCHEMBL9744042 0.82 NR1I2 (0.54) KDM4ENR1I2MAPTSLC22A6SLC22A8
Trifluoroacetic Acid SCHEMBL9878470 0.81 NR1I2 (0.59) NR1I2MAPTSLC22A6SLC22A8SLC22A11
SCHEMBL13576357 0.80 NR1I2 (0.60) NR1I2MAPTSLC22A6SLC22A8SLC22A11
SCHEMBL9744018 0.79 KDM4E (0.50) KDM4ENR1I2MAPTSLC22A6SLC22A8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5147871-A Anti-bacterial cephalosporin compounds HOFFMANN LA-ROCHE, INC. (US) 1992-09-15 US disclosed