SCHEMBL9747188

SCHEMBL9747188

Cn1c(N)c(N)c(=O)n(C)c1=S

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CASP6 P55212 1/20 0.59
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
KDM4A O75164 1/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL88218 0.75 ALDH1A1 (0.47) MAPTKDM4EALDH1A1POLBCYP2C19
Water SCHEMBL3902406 0.73 ALDH1A1 (0.46) MAPTKDM4EALDH1A1POLBCYP2C19
Hydrochloric Acid SCHEMBL6316692 0.73 ALDH1A1 (0.46) MAPTKDM4EALDH1A1POLBCYP2C19
Sulfurous Acid SCHEMBL5098561 0.67 ALDH1A1 (0.44) MAPTKDM4EALDH1A1POLBKMT2A
SCHEMBL3056710 0.64 ALDH1A1 (0.34) KDM4EALDH1A1POLBKMT2A
SCHEMBL33658 0.64 BCHE (0.33) CASP6KMT2A
SCHEMBL14791110 0.63 CASP6 (0.41) CASP6MAPTKDM4EKDM4AALDH1A1
SCHEMBL7473943 0.62 GSK3B (0.38) CASP6MAPTKDM4EALDH1A1POLB
SCHEMBL28438188 0.62 ADORA2A (0.45) MAPTKDM4EALDH1A1POLBCYP2C19
SCHEMBL28429328 0.62 TSHR (0.46) MAPTKDM4EALDH1A1POLBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0203721-B1 8-PHENYL XANTHINES THE WELLCOME FOUNDATION LIMITED (GB) 1992-06-10 EP disclosed
US-5017577-A Using Purine Cinnamic Acids BURROUGHS WELLCOME CO. (US) 1991-05-21 US disclosed
US-5015647-A Using Purine Cinnamic Acid Compounds BURROUGHS WELLCOME CO. (US) 1991-05-14 US disclosed
US-4981857-A ADENOSINE ANTAGONIST BURROUGHS WELLCOME CO. (US) 1991-01-01 US disclosed
US-4879296-A BLOCKING ADERNOSINE CELL SURFACE EFFECTS BURROUGHS WELLCOME CO. (US) 1989-11-07 US disclosed
EP-0203721-A2 8-Phenyl xanthines THE WELLCOME FOUNDATION LIMITED (GB) 1986-12-03 EP disclosed