SCHEMBL9748969

SCHEMBL9748969

O=C(NC(=O)c1ccc2ncccc2c1)NC1CCN(Cc2cc(O)ccc2O)CC1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 2/20 0.52
DRD4 P21917 6/20 0.49
CXCR4 P61073 1/20 0.48
HTR3A P46098 1/20 0.46
CCR3 P51677 4/20 0.45
PLK1 P53350 1/20 0.44
SLC6A12 P48065 1/20 0.44
SLC6A13 Q9NSD5 1/20 0.44
MCHR1 Q99705 1/20 0.44
DRD2 P14416 2/20 0.43
HTR2A P28223 2/20 0.43
DRD3 P35462 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9748761 0.85 ACKR3 (0.61) ACKR3DRD4CXCR4CCR3SLC6A12
SCHEMBL9748562 0.82 DRD4 (0.61) ACKR3DRD4SLC6A12SLC6A13MCHR1
SCHEMBL9748813 0.79 CCR3 (0.62) ACKR3DRD4CCR3MCHR1
SCHEMBL9589358 0.79 DRD4 (0.67) ACKR3DRD4CXCR4CCR3SLC6A12
SCHEMBL9592513 0.77 CXCR4 (0.61) ACKR3DRD4CXCR4CCR3MCHR1
SCHEMBL9750306 0.76 PLK1 (0.56) ACKR3HTR3APLK1
SCHEMBL9591604 0.71 DRD4 (0.65) DRD4SLC6A12MCHR1DRD2DRD3
SCHEMBL9591681 0.70 DRD4 (0.61) ACKR3DRD4CCR3MCHR1DRD2
SCHEMBL10530618 0.69 ADRA2A (0.69) DRD4CXCR4HTR3ADRD2HTR2A
SCHEMBL17270267 0.68 ACKR3 (1.00) ACKR3CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0234098-B1 N-[piperidylaminocarbonyl]quinolinecarboxamide derivatives having psychotropic activity JOHN WYETH & BROTHER LIMITED (GB) 1992-02-26 EP claimed