SCHEMBL9749134

SCHEMBL9749134

O=C(O)CC/C=C/c1ccc2ccccc2c1O

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.45
CYP1B1 Q16678 5/20 0.43
CYP1A1 P04798 4/20 0.43
ABCG2 Q9UNQ0 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
CFTR P13569 1/20 0.40
PTPN22 Q9Y2R2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9749139 1.00 LDHA (0.45) LDHACYP1B1CYP1A1ABCG2KDM4E
SCHEMBL9614832 0.81 TNF (0.44) KDM4EALDH1A1HPGD
SCHEMBL9614833 0.81 TNF (0.44) KDM4EALDH1A1HPGD
SCHEMBL765996 0.76 CYP1B1 (0.54) LDHACYP1B1CYP1A1ABCG2KDM4E
SCHEMBL765995 0.76 CYP1B1 (0.54) LDHACYP1B1CYP1A1ABCG2KDM4E
SCHEMBL10993947 0.75 SMPD2 (0.52) CYP1B1CYP1A1ALDH1A1HPGDCYP1A2
SCHEMBL10993939 0.75 SMPD2 (0.52) CYP1B1CYP1A1ALDH1A1HPGDCYP1A2
SCHEMBL9574440 0.74 NFKB1 (0.55) KDM4EALDH1A1
SCHEMBL9748807 0.74 GRIK1 (0.53) LDHACYP1B1CYP1A1ABCG2KDM4E
SCHEMBL9748809 0.74 GRIK1 (0.53) LDHACYP1B1CYP1A1ABCG2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0201071-B1 2-SUBSTITUTED-1-NAPHTHOLS AS 5-LIPOXYGENASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1992-03-04 EP claimed