SCHEMBL9748807

SCHEMBL9748807

CCC(C/C=C/c1ccc2ccccc2c1O)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 6/20 0.53
GRIK2 Q13002 6/20 0.53
SMPD2 O60906 2/20 0.43
GRIK3 Q13003 2/20 0.42
LDHA P00338 1/20 0.40
CYP1B1 Q16678 2/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP1A1 P04798 1/20 0.38
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9748809 1.00 GRIK1 (0.53) GRIK1GRIK2SMPD2GRIK3LDHA
SCHEMBL1716930 0.74 GRIK1 (0.65) GRIK1GRIK2GRIK3
SCHEMBL1716932 0.74 GRIK1 (0.65) GRIK1GRIK2GRIK3
SCHEMBL9749492 0.74 PPARG (0.46) LDHA
SCHEMBL9749139 0.74 LDHA (0.45) LDHACYP1B1ABCG2KDM4ECYP1A1
SCHEMBL9749134 0.74 LDHA (0.45) LDHACYP1B1ABCG2KDM4ECYP1A1
SCHEMBL9750303 0.74 ALDH1A1 (0.45) CYP1B1ABCG2KDM4EMEN1MAPT
SCHEMBL9750296 0.74 ALDH1A1 (0.45) CYP1B1ABCG2KDM4EMEN1MAPT
SCHEMBL765996 0.71 CYP1B1 (0.54) LDHACYP1B1ABCG2KDM4ECYP1A1
SCHEMBL765995 0.71 CYP1B1 (0.54) LDHACYP1B1ABCG2KDM4ECYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0201071-B1 2-SUBSTITUTED-1-NAPHTHOLS AS 5-LIPOXYGENASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1992-03-04 EP claimed